SCHEMBL4359730

SCHEMBL4359730

CC(C)(C)N(C[C@H](N)Cc1ccc(Cl)cc1)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.50
SLC6A2 P23975 1/20 0.44
SLC6A3 Q01959 1/20 0.44
CYP3A4 P08684 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
NFKB1 P19838 1/20 0.42
CYP2C19 P33261 1/20 0.42
LMNA P02545 2/20 0.41
PMP22 Q01453 1/20 0.41
NLRP3 Q96P20 1/20 0.41
DPP4 P27487 1/20 0.40
DPP7 Q9UHL4 1/20 0.40
PPARG P37231 2/20 0.39
PPARA Q07869 2/20 0.39
ANPEP P15144 2/20 0.38
ENPEP Q07075 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4359724 1.00 SLC6A4 (0.50) SLC6A4SLC6A2SLC6A3CYP3A4CYP1A2
SCHEMBL14860143 0.87 EPHX1 (0.48) LMNAANPEPALDH1A1HTTRAB9A
SCHEMBL14860145 0.87 EPHX1 (0.48) LMNAANPEPALDH1A1HTTRAB9A
SCHEMBL1527219 0.87 EPHX1 (0.48) LMNAANPEPALDH1A1HTTRAB9A
SCHEMBL4343817 0.86 RIPK1 (0.40) DPP4DPP7ANPEPENPEP
SCHEMBL4343822 0.86 RIPK1 (0.40) DPP4DPP7ANPEPENPEP
SCHEMBL4344087 0.85 PNMT (0.48) SLC6A4SLC6A2SLC6A3DPP4DPP7
SCHEMBL4344081 0.85 PNMT (0.48) SLC6A4SLC6A2SLC6A3DPP4DPP7
SCHEMBL4349347 0.84 LDHA (0.53) SLC6A4CYP1A2CYP2D6CYP2C19PPARG
SCHEMBL4349354 0.84 LDHA (0.53) SLC6A4CYP1A2CYP2D6CYP2C19PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2070928-A1 7-azaindol-3-ylacrylamides active as kinase inhibitors NERVIANO MEDICAL SCIENCES S.r.l. (IT) 2009-06-17 EP disclosed