SCHEMBL3777016

SCHEMBL3777016

COc1ccc(C[C@@H](CN)CN(C(=O)O)C(C)(C)C)cc1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.52
SLC6A4 P31645 1/20 0.41
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
TAS2R14 Q9NYV8 1/20 0.39
POLB P06746 1/20 0.39
ACHE P22303 1/20 0.39
APLNR P35414 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4349354 0.85 LDHA (0.53) LDHASLC6A4PPARGPPARACYP1A2
SCHEMBL4349347 0.85 LDHA (0.53) LDHASLC6A4PPARGPPARACYP1A2
SCHEMBL2209892 0.77 HTT (0.51) LDHATDP1TAS2R14ACHEAPLNR
SCHEMBL2293591 0.76 FFAR1 (0.43) PPARGPPARA
SCHEMBL14860429 0.76 CYP1A2 (0.46) LDHACYP1A2CYP2D6CYP2C19TDP1
SCHEMBL1025521 0.74 ALOX5 (0.52) LDHATAS2R14ACHE
SCHEMBL3777021 0.72 LDHA (0.49) LDHASLC6A4PPARGPPARACYP1A2
SCHEMBL14860143 0.71 EPHX1 (0.48)
SCHEMBL14860145 0.71 EPHX1 (0.48)
SCHEMBL1527219 0.71 EPHX1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100317697-A1 Renin Inhibitors VITAE PHARMACEUTICALS, INC. 2010-12-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100317697-A1 Renin Inhibitors REN, ACE, SERPINB1 LDHA 843/4885SLC6A4 2399/4885PPARG 3070/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.