SCHEMBL4351653

SCHEMBL4351653

Oc1c(F)cc(NCc2ccccc2Sc2cccc(Cl)c2)cc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 4/20 0.53
SLC6A2 P23975 2/20 0.53
SLC6A3 Q01959 2/20 0.53
CYP2C9 P11712 3/20 0.46
CYP2C19 P33261 3/20 0.46
CYP1A2 P05177 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
CYP3A4 P08684 2/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALOX15 P16050 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PLA2G1B P04054 1/20 0.41
CYP2D6 P10635 1/20 0.41
ATG4B Q9Y4P1 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4354072 0.88 SLC6A2 (0.48) SLC6A4SLC6A2SLC6A3CYP2C9CYP2C19
SCHEMBL4354940 0.88 SLC6A4 (0.52) SLC6A4SLC6A2SLC6A3CYP2C9CYP2C19
SCHEMBL4347073 0.88 MEN1 (0.49) SLC6A4SLC6A2SLC6A3CYP2C9CYP2C19
SCHEMBL4345358 0.88 MAPT (0.47) SLC6A4SLC6A2SLC6A3CYP2C9CYP2C19
SCHEMBL4354639 0.87 LMNA (0.44) SLC6A4SLC6A2SLC6A3CYP2C9CYP2C19
SCHEMBL4354085 0.87 SLC6A4 (0.51) SLC6A4SLC6A2SLC6A3CYP2C9CYP2C19
SCHEMBL4342244 0.86 MEN1 (0.50) SLC6A4SLC6A2SLC6A3CYP2C9CYP2C19
SCHEMBL4351152 0.86 SLC6A4 (0.50) SLC6A4SLC6A2SLC6A3CYP2C9CYP2C19
SCHEMBL4359801 0.85 SLC6A4 (0.49) SLC6A4SLC6A2SLC6A3CYP2C9CYP2C19
SCHEMBL12846505 0.84 SLC6A4 (0.51) SLC6A4SLC6A2SLC6A3CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed