SCHEMBL4354639

SCHEMBL4354639

Oc1c(F)cc(NCc2ccccc2Sc2ccccc2)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
CHRNA7 P36544 2/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
GAA P10253 1/20 0.41
APOBEC3A P31941 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
MAOB P27338 1/20 0.40
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4350004 0.90 MAPT (0.46) LMNASMN1; SMN2CYP1A2CYP2C9CYP2C19
SCHEMBL4347073 0.90 MEN1 (0.49) LMNASMN1; SMN2CYP1A2CYP2C9CYP2C19
SCHEMBL4351653 0.87 SLC6A4 (0.53) LMNASMN1; SMN2CYP1A2CYP2C9CYP2C19
SCHEMBL4346787 0.86 NOX4 (0.45) LMNASMN1; SMN2CYP1A2CYP2C9CYP2C19
SCHEMBL4359446 0.86 MEN1 (0.58) LMNACYP2C9CYP2C19L3MBTL1SLC6A2
SCHEMBL4345667 0.86 ALDH3A1 (0.50) LMNASMN1; SMN2L3MBTL1ALDH1A1HPGD
SCHEMBL4342244 0.85 MEN1 (0.50) LMNASMN1; SMN2CYP1A2CYP2C9CYP2C19
SCHEMBL4352975 0.84 GPR39 (0.41) LMNASMN1; SMN2L3MBTL1ALDH1A1SLC6A2
SCHEMBL4347830 0.84 ALDH3A1 (0.46) LMNASMN1; SMN2ALDH1A1GAAMAOB
SCHEMBL4347048 0.84 CYP2C9 (0.47) LMNACYP1A2CYP2C9CYP2C19L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed