SCHEMBL4358260

SCHEMBL4358260

CC(C)(C)N(S)C(=O)Nc1cc(Br)cc(F)c1O

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.34
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
ALDH1A1 P00352 2/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
GAA P10253 1/20 0.31
GPR35 Q9HC97 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
ACLY P53396 1/20 0.30
PDK1 Q15118 1/20 0.30
PDK2 Q15119 1/20 0.30
PDK3 Q15120 1/20 0.30
PDK4 Q16654 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12362248 0.79 PDK1 (0.39) HTTKDM4ENPC1RAB9AALDH1A1
SCHEMBL4346269 0.78 CXCR2 (0.39) HTTKDM4ENPC1RAB9AALDH1A1
SCHEMBL4353361 0.77 XDH (0.39) HTTALDH1A1GAA
SCHEMBL4354426 0.77 NPC1 (0.47) HTTKDM4ENPC1RAB9AALDH1A1
SCHEMBL4346777 0.75 HTT (0.38) HTTKDM4ENPC1ALDH1A1LMNA
SCHEMBL16654497 0.75 NPC1 (0.41) HTTNPC1RAB9AALDH1A1LMNA
SCHEMBL27761067 0.73 KIF11 (0.47) HTTNPC1RAB9AALDH1A1LMNA
SCHEMBL4343499 0.73 ALDH1A1 (0.39) HTTKDM4EALDH1A1LMNAGAA
SCHEMBL4342070 0.72 EGFR (0.43) NPC1RAB9AALDH1A1LMNASMN1; SMN2
SCHEMBL4343991 0.71 HTT (0.40) HTTNPC1RAB9AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
US-20070054904-A1 Phenol derivatives and their use as rotamase inhibitors JERINI AG (DE) 2007-03-08 US claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070054904-A1 Phenol derivatives and their use as rotamase inhibitors NR1I3, NR1D1, NR1D2 HTT 3995/4885KDM4E 1689/4885NPC1 1189/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.