SCHEMBL4350068

SCHEMBL4350068

O=C(NCc1ccc(C(F)(F)F)cc1)Nc1cc(Br)c(O)c(Br)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 4/20 0.67
NAMPT P43490 2/20 0.60
PRMT3 O60678 1/20 0.54
TRPV1 Q8NER1 3/20 0.52
CNR1 P21554 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
MCHR1 Q99705 1/20 0.47
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
EPHX2 P34913 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4348348 0.85 MTOR (0.69) MTORNAMPTPRMT3TRPV1CNR1
SCHEMBL4353993 0.84 MTOR (0.67) MTORNAMPTPRMT3TRPV1CNR1
SCHEMBL4351636 0.84 MEN1 (0.61) MTORMEN1KMT2ALMNASMN1; SMN2
SCHEMBL4348910 0.83 EPHX2 (0.69) MTORTRPV1MEN1KMT2ASMN1; SMN2
SCHEMBL4347380 0.82 CA1 (0.56) NAMPTMEN1KMT2ASMN1; SMN2CA1
SCHEMBL28808075 0.79 MTOR (0.76) MTORNAMPTPRMT3MEN1KMT2A
SCHEMBL26625460 0.79 MTOR (0.71) MTORNAMPTPRMT3TRPV1MEN1
SCHEMBL6668636 0.79 MTOR (0.48) MTORNAMPTCNR1MCHR1EPHX2
SCHEMBL4347646 0.78 MTOR (0.70) MTORNAMPTPRMT3TRPV1CNR1
SCHEMBL24575984 0.78 MTOR (0.69) MTORNAMPTPRMT3TRPV1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed