SCHEMBL4354053

SCHEMBL4354053

CCCCCNC(=O)N(S)c1cc(F)c(O)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.44
EPHX2 P34913 1/20 0.43
EPHX1 P07099 6/20 0.42
NAAA Q02083 3/20 0.42
LMNA P02545 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPK3 P27361 1/20 0.40
ASAH1 Q13510 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SQOR Q9Y6N5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4350102 0.87 TRPV1 (0.49) TRPV1EPHX2NAAA
SCHEMBL4350363 0.84 TRPV1 (0.43) TRPV1EPHX1NAAAASAH1
SCHEMBL4348484 0.84 EPHX2 (0.43) TRPV1EPHX2EPHX1NAAA
SCHEMBL4349401 0.80 MGLL (0.38) TRPV1EPHX2EPHX1NAAALMNA
SCHEMBL4350070 0.79 NAAA (0.40) TRPV1EPHX2EPHX1NAAASMN1; SMN2
SCHEMBL4355852 0.79 EPHX2 (0.48) TRPV1EPHX2EPHX1NAAALMNA
SCHEMBL4351425 0.76 EPHX2 (0.37) TRPV1EPHX2EPHX1NAAA
SCHEMBL4346130 0.76 CA1 (0.51) TRPV1EPHX2EPHX1NAAA
SCHEMBL4349030 0.75 RAB9A (0.49) TRPV1EPHX1
SCHEMBL4358550 0.74 EPHX2 (0.39) TRPV1EPHX2EPHX1NAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed