SCHEMBL4354896

SCHEMBL4354896

COc1cnc2cc(I)c(C(=O)N3CC4(C)CN(C(=O)c5cc6nc(OC)cnc6cc5I)CC(C)(C3)C4)cc2n1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.34
PDGFRB P09619 2/20 0.33
PDGFRA P16234 2/20 0.33
HCRTR1 O43613 6/20 0.33
HCRTR2 O43614 6/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
AVPR2 P30518 1/20 0.31
AVPR1A P37288 1/20 0.31
PIK3CD O00329 2/20 0.30
PIK3CA P42336 2/20 0.30
PIK3CG P48736 2/20 0.30
PIK3CB P42338 1/20 0.30
SIRT6 Q8N6T7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4342604 0.89 GAA (0.39) HPGDPDGFRBPDGFRAHCRTR1HCRTR2
SCHEMBL4350380 0.74 FASN (0.34) HCRTR1HCRTR2
SCHEMBL4349455 0.66 ALDH1A1 (0.33)
SCHEMBL4354630 0.65 PDE2A (0.33) HPGD
SCHEMBL4341690 0.64 ALDH1A1 (0.34)
SCHEMBL4350159 0.63 TSHR (0.34) HPGD
SCHEMBL14437924 0.61 PDGFRB (0.63) PDGFRBPDGFRA
SCHEMBL4346476 0.61 HPGD (0.61) HPGD
SCHEMBL4351695 0.61 KDM4E (0.49) HPGD
SCHEMBL719716 0.60 MAOA (0.44) PDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2088149-A1 PHARMACOLOGICALLY ACTIVE N,N'-SUBSTITUTED 3,7-DIAZABICYCLO Ý3.3.1¨NONANES, PHARMACEUTICAL COMPOSITIONS BASED THEREON AND A METHOD FOR THE USE THEREOF Institute of Physiologically active compunds of the Russian Academy of Sciences (IPAC RAN) (RU) 2009-08-12 EP claimed
EP-2088149-A1 PHARMACOLOGICALLY ACTIVE N,N'-SUBSTITUTED 3,7-DIAZABICYCLO Ý3.3.1¨NONANES, PHARMACEUTICAL COMPOSITIONS BASED THEREON AND A METHOD FOR THE USE THEREOF Institute of Physiologically active compunds of the Russian Academy of Sciences (IPAC RAN) (RU) 2009-08-12 EP disclosed