SCHEMBL4355970

SCHEMBL4355970

CN1CCN(C2(CNC(=O)c3cn(-c4ncccn4)c4cccc(F)c34)CCCCC2)CC1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCN1 O60741 7/20 0.54
HCN4 Q9Y3Q4 6/20 0.53
TP53 P04637 3/20 0.52
OPRM1 P35372 2/20 0.49
SIGMAR1 Q99720 2/20 0.49
THRB P10828 3/20 0.47
LMNA P02545 3/20 0.47
SLC6A9 P48067 1/20 0.46
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
P2RX7 Q99572 1/20 0.45
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4353725 0.92 HCN4 (0.54) HCN1HCN4TP53SLC6A9ALDH1A1
SCHEMBL4350496 0.91 HCN4 (0.55) HCN1HCN4TP53SLC6A9ALDH1A1
SCHEMBL4355954 0.90 HCN1 (0.62) HCN1HCN4TP53OPRM1SIGMAR1
SCHEMBL3688404 0.90 HCN4 (0.63) HCN1HCN4TP53OPRM1SIGMAR1
SCHEMBL4357339 0.90 HCN4 (0.63) HCN1HCN4TP53OPRM1SIGMAR1
SCHEMBL4359934 0.89 HCN1 (0.42) HCN1HCN4TP53OPRM1SIGMAR1
SCHEMBL13706728 0.89 HCN1 (0.42) HCN1HCN4TP53OPRM1SIGMAR1
SCHEMBL4351759 0.87 HCN4 (0.60) HCN1HCN4TP53OPRM1SIGMAR1
SCHEMBL4358058 0.85 HCN1 (0.42) HCN1HCN4LMNASLC6A9ALDH1A1
SCHEMBL13706822 0.85 HCN1 (0.42) HCN1HCN4LMNASLC6A9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009108551-A2 HETEROARYL AMIDE ANALOGUES H. LUNDBECK A/S (DK) 2009-09-03 WO claimed
WO-2009108551-A2 HETEROARYL AMIDE ANALOGUES H. LUNDBECK A/S (DK) 2009-09-03 WO disclosed