SCHEMBL4358300

SCHEMBL4358300

CCOC(=O)CCNC(=O)Nc1ccc(O)c(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.52
MAPT P10636 5/20 0.52
HSD17B10 Q99714 4/20 0.52
HPGD P15428 4/20 0.52
KDM4E B2RXH2 3/20 0.52
HTT P42858 3/20 0.52
PTPN7 P35236 1/20 0.52
NPSR1 Q6W5P4 3/20 0.52
LMNA P02545 3/20 0.52
MAPK1 P28482 2/20 0.52
EPHX2 P34913 4/20 0.51
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
GAA P10253 2/20 0.48
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
RORC P51449 1/20 0.44
CASR P41180 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4345924 0.86 ALDH1A1 (0.52) ALDH1A1MAPTHSD17B10HPGDKDM4E
SCHEMBL6229381 0.85 ALDH1A1 (0.54) ALDH1A1MAPTHSD17B10HPGDKDM4E
SCHEMBL4359582 0.85 ALDH1A1 (0.52) ALDH1A1MAPTHSD17B10HPGDKDM4E
SCHEMBL4346283 0.81 ALDH1A1 (0.49) ALDH1A1MAPTHSD17B10HPGDKDM4E
SCHEMBL15741795 0.81 ALDH1A1 (0.66) ALDH1A1HSD17B10HPGDLMNAMAPK1
SCHEMBL27761103 0.80 EPHX2 (0.67) ALDH1A1MAPTHTTEPHX2MEN1
SCHEMBL4349661 0.80 MEN1 (0.67) ALDH1A1MAPTHSD17B10HPGDKDM4E
SCHEMBL4348602 0.79 EPHX2 (0.74) ALDH1A1MAPTHTTEPHX2MEN1
SCHEMBL6230978 0.78 ALDH1A1 (0.45) ALDH1A1MAPTHSD17B10HPGDKDM4E
SCHEMBL4359586 0.78 ALDH1A1 (0.45) ALDH1A1MAPTHSD17B10HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed