SCHEMBL4346283

SCHEMBL4346283

CCOC(=O)CCNC(=O)Nc1ccc(O)c([N+](=O)[O-])c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.49
PTPN7 P35236 1/20 0.48
MAPT P10636 9/20 0.46
KDM4E B2RXH2 4/20 0.46
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
LMNA P02545 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
USP2 O75604 1/20 0.45
MAPK1 P28482 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
HSD17B10 Q99714 3/20 0.44
NPSR1 Q6W5P4 3/20 0.44
HTT P42858 4/20 0.43
HPGD P15428 2/20 0.43
SLC6A3 Q01959 1/20 0.43
BCL6 P41182 1/20 0.42
BCOR Q6W2J9 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6670113 0.94 ALDH1A1 (0.51) ALDH1A1PTPN7MAPTKDM4EHTT
SCHEMBL27782790 0.82 EPHX1 (0.50) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL4358300 0.81 ALDH1A1 (0.52) ALDH1A1PTPN7MAPTKDM4EMEN1
SCHEMBL4354492 0.81 EPHX1 (0.55) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL4359582 0.81 ALDH1A1 (0.52) ALDH1A1PTPN7MAPTKDM4EMEN1
SCHEMBL8601321 0.80 EPHX1 (0.57) ALDH1A1MAPTHTTSLC6A3
SCHEMBL8598927 0.80 EPHX1 (0.57) ALDH1A1MAPTHTTSLC6A3
SCHEMBL8194387 0.77 MAPT (0.58) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL4351840 0.75 CA2 (0.59) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL6966529 0.75 MAPT (0.53) ALDH1A1MAPTKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed