SCHEMBL4358617

SCHEMBL4358617

Cc1ccccc1CNC(=S)Nc1ccc(O)c(F)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.52
LMNA P02545 5/20 0.52
MEN1 O00255 5/20 0.52
KMT2A Q03164 5/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
PKM P14618 1/20 0.52
CRHBP P24387 1/20 0.52
CRHR2 Q13324 1/20 0.52
HTT P42858 1/20 0.50
ALDH1A1 P00352 2/20 0.49
MAPK1 P28482 1/20 0.47
ALOX12 P18054 2/20 0.45
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
POLB P06746 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
HDAC1 Q13547 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4345586 0.87 LMNA (0.51) MAPTLMNAMEN1KMT2ASMN1; SMN2
SCHEMBL4341716 0.85 RAB9A (0.62) MEN1KMT2APKMALDH1A1MAPK1
SCHEMBL4357807 0.85 MAPT (0.54) MAPTLMNAMEN1KMT2ASMN1; SMN2
SCHEMBL4343714 0.81 RAB9A (0.63) MAPTLMNAMEN1KMT2ASMN1; SMN2
SCHEMBL4347021 0.80 MEN1 (0.64) MAPTLMNAMEN1KMT2ASMN1; SMN2
SCHEMBL4358359 0.76 SMN1; SMN2 (0.45) MAPTLMNAMEN1KMT2ASMN1; SMN2
SCHEMBL4348819 0.76 MEN1 (0.54) MAPTLMNAMEN1KMT2ASMN1; SMN2
SCHEMBL4349842 0.75 KMT2A (0.56) MAPTLMNAMEN1KMT2ASMN1; SMN2
SCHEMBL6226788 0.75 LMNA (0.54) MAPTLMNAMEN1KMT2ASMN1; SMN2
SCHEMBL4351089 0.74 LMNA (0.64) MAPTLMNAMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed