SCHEMBL4345586

SCHEMBL4345586

Cc1ccccc1CNC(=S)Nc1cc(F)c(O)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 6/20 0.51
MAPT P10636 5/20 0.51
SMN1; SMN2 Q16637 5/20 0.51
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
PKM P14618 1/20 0.51
CRHBP P24387 1/20 0.51
CRHR2 Q13324 1/20 0.51
HTT P42858 3/20 0.49
ALDH1A1 P00352 4/20 0.48
POLB P06746 2/20 0.45
ALOX12 P18054 3/20 0.44
MAPK1 P28482 1/20 0.43
MAOB P27338 1/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4358617 0.87 MAPT (0.52) LMNAMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL4348819 0.84 MEN1 (0.54) LMNAMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL4342163 0.84 RAB9A (0.61) MAPTMEN1KMT2APKMHTT
SCHEMBL4358359 0.84 SMN1; SMN2 (0.45) LMNAMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL4345595 0.81 MEN1 (0.46) LMNAMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL4345336 0.80 MAOB (0.66) LMNAMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL4349842 0.80 KMT2A (0.56) LMNAMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL4354182 0.79 ALOX12 (0.51) LMNAMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL4357807 0.76 MAPT (0.54) LMNAMAPTSMN1; SMN2MEN1KMT2A
SCHEMBL4345459 0.76 MEN1 (0.46) LMNAMAPTSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed