SCHEMBL4358359

SCHEMBL4358359

Cc1ccccc1CNC(=S)Nc1cc(Br)c(O)c(Br)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.45
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
ALOX12 P18054 5/20 0.44
MAPT P10636 5/20 0.44
LMNA P02545 4/20 0.44
ALDH1A1 P00352 5/20 0.43
HTT P42858 2/20 0.43
HPGD P15428 2/20 0.43
POLB P06746 1/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4345586 0.84 LMNA (0.51) SMN1; SMN2MEN1KMT2AALOX12MAPT
SCHEMBL4348819 0.84 MEN1 (0.54) SMN1; SMN2MEN1KMT2AALOX12MAPT
SCHEMBL4345433 0.80 MAOB (0.66) SMN1; SMN2MEN1KMT2AALOX12MAPT
SCHEMBL4358617 0.76 MAPT (0.52) SMN1; SMN2MEN1KMT2AALOX12MAPT
SCHEMBL4357807 0.76 MAPT (0.54) SMN1; SMN2MEN1KMT2AALOX12MAPT
SCHEMBL4345595 0.76 MEN1 (0.46) SMN1; SMN2MEN1KMT2AALOX12MAPT
SCHEMBL4345459 0.76 MEN1 (0.46) SMN1; SMN2MEN1KMT2AALOX12MAPT
SCHEMBL4349820 0.73 ALOX12 (0.56) SMN1; SMN2MEN1KMT2AALOX12MAPT
SCHEMBL4347019 0.73 ALOX12 (0.59) SMN1; SMN2MEN1KMT2AALOX12MAPT
SCHEMBL4355354 0.73 ALDH1A1 (0.63) SMN1; SMN2MEN1KMT2AALOX12MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed