SCHEMBL4362296

SCHEMBL4362296

C[C@@H](Nc1c(NC2CCNCC2)c(=O)c1=O)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.48
CYP2C9 P11712 2/20 0.48
MAPKAPK2 P49137 9/20 0.48
AURKB Q96GD4 3/20 0.48
MAPK1 P28482 3/20 0.48
ROCK1 Q13464 2/20 0.48
PLK1 P53350 2/20 0.48
PDGFRA P16234 2/20 0.48
CSNK1G1 Q9HCP0 2/20 0.48
DCLK1 O15075 1/20 0.48
ROCK2 O75116 1/20 0.48
CHEK2 O96017 1/20 0.48
GSK3A P49840 1/20 0.48
GSK3B P49841 1/20 0.48
IRAK1 P51617 1/20 0.48
PRKX P51817 1/20 0.48
NEK4 P51957 1/20 0.48
CSNK1G2 P78368 1/20 0.48
CDC42BPA Q5VT25 1/20 0.48
BRSK1 Q8TDC3 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4560397 0.92 CXCR2 (0.44) CYP3A4CYP2C9MAPKAPK2AURKBMAPK1
SCHEMBL4378340 0.79 HTT (0.50) CYP3A4CYP2C9MAPKAPK2AURKBMAPK1
SCHEMBL4153139 0.75 GAA (0.71) MAPK1SOS1GAAL3MBTL1
SCHEMBL4371405 0.74 ALDH1A1 (0.58) MAPK1GAAL3MBTL1
SCHEMBL17920542 0.70 MAPKAPK2 (0.80) CYP3A4CYP2C9MAPKAPK2AURKBMAPK1
SCHEMBL4374908 0.68 MAPKAPK2 (0.55) CYP3A4CYP2C9MAPKAPK2AURKBMAPK1
SCHEMBL6009184 0.66 GRM7 (0.64) CYP3A4SOS1
SCHEMBL11390159 0.66 RECQL (0.75) GAA
SCHEMBL27787057 0.66 HPGD (0.77) CYP3A4SOS1
SCHEMBL918020 0.65 HTR6 (0.49) SOS1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009012375-A2 SQUARATE KINASE INHIBITORS WYETH (US) 2009-01-22 WO disclosed