SCHEMBL4378340

SCHEMBL4378340

C[C@@H](Nc1c(NC2CC(C)(C)NC(C)(C)C2)c(=O)c1=O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.50
POLB P06746 1/20 0.49
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
PKM P14618 1/20 0.47
ALOX15 P16050 1/20 0.47
ALOX12 P18054 1/20 0.47
RAD52 P43351 1/20 0.47
GFER P55789 1/20 0.47
KMT2A Q03164 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 2/20 0.46
MAPKAPK2 P49137 5/20 0.46
ROCK1 Q13464 2/20 0.46
AURKB Q96GD4 2/20 0.46
DCLK1 O15075 1/20 0.46
ROCK2 O75116 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4362296 0.79 CYP3A4 (0.48) L3MBTL1CYP3A4CYP2C9MAPKAPK2ROCK1
SCHEMBL9668473 0.76 GAA (0.57) HTTPOLBALDH1A1MEN1LMNA
Trifluoroacetic Acid SCHEMBL4560397 0.72 CXCR2 (0.44) LMNACYP3A4CYP2C9MAPKAPK2ROCK1
SCHEMBL9380274 0.69 KMT2A (0.87) HTTPOLBALDH1A1MEN1LMNA
SCHEMBL17920542 0.68 MAPKAPK2 (0.80) CYP3A4CYP2C9MAPKAPK2ROCK1AURKB
SCHEMBL4371405 0.68 ALDH1A1 (0.58) HTTALDH1A1MEN1LMNAMAPT
SCHEMBL15613273 0.67 HTT (1.00) HTTPOLBMEN1MAPTKMT2A
SCHEMBL4374908 0.67 MAPKAPK2 (0.55) MEN1KMT2ACYP3A4CYP2C9MAPKAPK2
SCHEMBL3225224 0.66 MEN1 (0.51) POLBALDH1A1MEN1LMNAMAPT
SCHEMBL27991724 0.66 POLB (0.50) HTTPOLBALDH1A1MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009012375-A2 SQUARATE KINASE INHIBITORS WYETH (US) 2009-01-22 WO claimed
WO-2009012375-A2 SQUARATE KINASE INHIBITORS WYETH (US) 2009-01-22 WO disclosed