SCHEMBL4363405

SCHEMBL4363405

O=C(c1cc2ccccc2n1CC(F)(F)F)N1CCOCC1Br

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.46
CNR2 P34972 5/20 0.37
PADI4 Q9UM07 2/20 0.35
CCR2 P41597 4/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
CNR1 P21554 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4366003 0.80 HRH3 (0.53) HRH3
SCHEMBL4365923 0.79 HRH3 (0.59) HRH3PADI4
SCHEMBL3539771 0.70 HRH3 (0.63) HRH3PTGS1PTGS2
SCHEMBL2768671 0.68 HRH3 (0.64) HRH3CCR2PTGS1PTGS2
SCHEMBL3538545 0.67 HRH3 (0.71) HRH3PTGS1PTGS2
SCHEMBL23052993 0.66 NOD2 (0.64) CCR2
SCHEMBL4373527 0.65 HRH3 (0.44) HRH3CNR2
SCHEMBL3542210 0.63 HRH3 (1.00) HRH3CNR2
SCHEMBL3544224 0.62 HRH3 (0.95) HRH3CNR2
SCHEMBL30121932 0.62 ALDH1A1 (0.56) CNR2CCR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010487-A1 5-AMIDO-2-CARBOXAMIDE INDOLES F. Hoffmann-Roche AG (CH) 2009-01-07 EP disclosed
WO-2007115938-A1 5-AMIDO-2-CARBOXAMIDE INDOLES F. HOFFMANN-LA ROCHE AG (CH) 2007-10-18 WO disclosed