SCHEMBL4373527

SCHEMBL4373527

O=C(C1COCCN1C(=O)c1cc2ccccc2n1CC1CC1)N1CCN(C2CCCC2)CC1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.44
CNR2 P34972 1/20 0.41
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
ACACB O00763 3/20 0.39
ACACA Q13085 3/20 0.39
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
F10 P00742 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4365923 0.88 HRH3 (0.59) HRH3TMEM97SIGMAR1ACACBACACA
SCHEMBL4364219 0.83 SIGMAR1 (0.43) HRH3SIGMAR1ACACBACACAKDM4E
SCHEMBL3541201 0.75 HRH3 (0.74) HRH3CNR2ACACBACACA
SCHEMBL4366003 0.73 HRH3 (0.53) HRH3F10
SCHEMBL27760334 0.67 HRH3 (0.57) HRH3CNR2KDM4EALDH1A1
SCHEMBL3541739 0.67 HRH3 (0.57) HRH3CNR2KDM4EALDH1A1
SCHEMBL28306098 0.67 CCR2 (0.66) CNR2ALDH1A1
SCHEMBL3539042 0.67 HRH3 (0.59) HRH3KDM4EALDH1A1
SCHEMBL4361046 0.66 PROKR1 (0.43)
SCHEMBL3539590 0.66 HRH3 (0.60) HRH3CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010487-A1 5-AMIDO-2-CARBOXAMIDE INDOLES F. Hoffmann-Roche AG (CH) 2009-01-07 EP disclosed
WO-2007115938-A1 5-AMIDO-2-CARBOXAMIDE INDOLES F. HOFFMANN-LA ROCHE AG (CH) 2007-10-18 WO disclosed