SCHEMBL4371875

SCHEMBL4371875

COc1cc(Br)c2c(c1)CCCC2.Oc1cc(Br)c2c(c1)CCCC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.40
ALOX5 P09917 3/20 0.40
KIT P10721 4/20 0.36
PDGFRA P16234 4/20 0.36
FLT4 P35916 4/20 0.36
KDR P35968 4/20 0.36
FLT3 P36888 4/20 0.36
CYP3A4 P08684 2/20 0.36
CYP1A1 P04798 3/20 0.36
CYP1B1 Q16678 3/20 0.36
PDGFRB P09619 2/20 0.36
MAP2K1 Q02750 2/20 0.36
TTR P02766 2/20 0.36
MAP2K2 P36507 1/20 0.36
ALK Q9UM73 1/20 0.36
FLT1 P17948 1/20 0.36
KDM4E B2RXH2 5/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2999364 0.90 ALDH1A1 (0.39) CYP1A1CYP1B1MEN1KMT2AALDH1A1
SCHEMBL30550463 0.90 ALDH1A1 (0.39) CYP1A1CYP1B1MEN1KMT2AALDH1A1
SCHEMBL23731386 0.86 EGFR (0.40) CYP1A1CYP1B1ALDH1A1EGFRNPC1
SCHEMBL3002812 0.86 BCL2L1 (0.38) PTGS2ALOX5CYP3A4KDM4EGAA
SCHEMBL22618607 0.82 MAOA (0.37) PTGS2ALOX5CYP3A4KDM4EGAA
SCHEMBL29383596 0.82 MAOA (0.37) PTGS2ALOX5CYP3A4KDM4EGAA
SCHEMBL21357843 0.78 CYP3A4 (0.47) PTGS2ALOX5KITPDGFRAFLT4
SCHEMBL30777410 0.78 CYP3A4 (0.47) PTGS2ALOX5KITPDGFRAFLT4
SCHEMBL21584122 0.74 PTGS2 (0.34) PTGS2ALOX5ESR1BACE1
SCHEMBL2999085 0.74 PGR (0.47) CYP3A4TTRKDM4ESMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2070921-A1 Indolylmaleimide derivatives as protein kinase c inhibitors Novartis Ag (CH) 2009-06-17 EP disclosed