SCHEMBL4374753

SCHEMBL4374753

O=C(O)C[C@@H](c1ccc2c(c1)OCC2)N1CC[C@@H](CCCC2=CC=C3CCCNC3N2)C1=O

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 20/20 0.65
ITGAV P06756 20/20 0.65
ITGA2B P08514 2/20 0.34
ITGB1 P05556 1/20 0.34
ITGB6 P18564 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4379967 1.00 ITGB3 (0.65) ITGB3ITGAVITGA2BITGB1ITGB6
SCHEMBL4372614 0.91 ITGB3 (0.54) ITGB3ITGAVITGA2B
SCHEMBL4378958 0.91 ITGB3 (0.54) ITGB3ITGAVITGA2B
SCHEMBL4050199 0.88 ITGB3 (0.51) ITGB3ITGAV
SCHEMBL4370764 0.86 ITGB3 (0.48) ITGB3ITGAV
SCHEMBL4053563 0.85 ITGB3 (0.50) ITGB3ITGAV
SCHEMBL7553084 0.85 ITGAV (0.63) ITGB3ITGAVITGA2BITGB1ITGB6
SCHEMBL7595642 0.85 ITGAV (0.63) ITGB3ITGAVITGA2BITGB1ITGB6
SCHEMBL7592559 0.85 ITGAV (0.63) ITGB3ITGAVITGA2BITGB1ITGB6
SCHEMBL4374388 0.84 ITGB3 (0.45) ITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047425-A4 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2009-04-22 EP disclosed
EP-1047425-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-11-02 EP disclosed
WO-1999030709-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed