Alpha-Cyano-4-Hydroxycinnamic Acid

Alpha-Cyano-4-Hydroxycinnamic Acid

SCHEMBL437568

N#C/C(=C/c1ccc(O)cc1)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 1.00
ALDH1A1 P00352 2/20 1.00
CISD1 Q9NZ45 1/20 1.00
SLC16A3 O15427 1/20 1.00
CYP3A4 P08684 1/20 1.00
HPGD P15428 1/20 1.00
SLC16A1 P53985 1/20 1.00
GPR35 Q9HC97 1/20 1.00
EGFR P00533 3/20 0.73
MEN1 O00255 1/20 0.65
KMT2A Q03164 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alpha-Cyano-4-Hydroxycinnamic Acid SCHEMBL28529867 1.00 KDM4E (1.00) KDM4EALDH1A1CISD1SLC16A3CYP3A4
Alpha-Cyano-4-Hydroxycinnamic Acid SCHEMBL26826 1.00 KDM4E (1.00) KDM4EALDH1A1CISD1SLC16A3CYP3A4
Alpha-Cyano-4-Hydroxycinnamic Acid SCHEMBL26825 1.00 KDM4E (1.00) KDM4EALDH1A1CISD1SLC16A3CYP3A4
Alpha-Cyano-4-Hydroxycinnamic Acid SCHEMBL5530234 0.95 ALDH1A1 (0.90) KDM4EALDH1A1CISD1SLC16A3CYP3A4
Alpha-Cyano-4-Hydroxycinnamic Acid SCHEMBL5330094 0.93 KDM4E (0.87) KDM4EALDH1A1CISD1SLC16A3CYP3A4
Alpha-Cyano-4-Hydroxycinnamic Acid SCHEMBL5330088 0.93 KDM4E (0.87) KDM4EALDH1A1CISD1SLC16A3CYP3A4
SCHEMBL4600832 0.92 EGFR (0.85) KDM4EALDH1A1CISD1SLC16A3CYP3A4
SCHEMBL10413058 0.92 EGFR (0.85) KDM4EALDH1A1CISD1SLC16A3CYP3A4
SCHEMBL4600830 0.92 EGFR (0.85) KDM4EALDH1A1CISD1SLC16A3CYP3A4
Alpha-Cyano-4-Hydroxycinnamic Acid SCHEMBL28674225 0.92 ALDH1A1 (0.84) KDM4EALDH1A1CISD1SLC16A3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595952-B1 AGONISTS OF GPR40 CONNEXIOS LIFE SCIENCES PVT LTD (IN) 2020-11-18 EP disclosed
EP-2595952-B1 AGONISTS OF GPR40 CONNEXIOS LIFE SCIENCES PVT LTD (IN) 2020-11-18 EP disclosed
WO-2019078145-A1 MATERIAL FOR PREPARING MASS SPECTROMETRY SAMPLE JSR株式会社 2019-04-25 WO disclosed
US-9278915-B2 Agonists of GPR40 CONNEXIOS LIFE SCIENCES PVT LTD (IN) 2016-03-08 US disclosed
US-9278915-B2 Agonists of GPR40 CONNEXIOS LIFE SCIENCES PVT LTD (IN) 2016-03-08 US disclosed
US-9278915-B2 Agonists of GPR40 CONNEXIOS LIFE SCIENCES PVT LTD (IN) 2016-03-08 US disclosed
EP-2797886-A2 PAIN RELIEF COMPOUNDS Ecole Nationale Superieure de Chimie de Clermont Ferrand (FR) 2014-11-05 EP disclosed
US-20130237571-A1 AGONISTS OF GPR40 Conexios Life Sciences PVT. LTD. (IN) 2013-09-12 US disclosed
US-20130237571-A1 AGONISTS OF GPR40 Conexios Life Sciences PVT. LTD. (IN) 2013-09-12 US disclosed
US-20130237571-A1 AGONISTS OF GPR40 Conexios Life Sciences PVT. LTD. (IN) 2013-09-12 US disclosed
WO-2013098416-A2 PAIN RELIEF COMPOUNDS ECOLE NATIONALE SUPERIEURE DE CHIMIE DE CLERMONT FERRAND (FR) 2013-07-04 WO disclosed
EP-2595952-A1 AGONISTS OF GPR40 Connexios Life Sciences Pvt. Ltd. (IN) 2013-05-29 EP disclosed
WO-2012011125-A1 AGONISTS OF GPR40 CONNEXIOS LIFE SCIENCES PVT. LTD. (IN) 2012-01-26 WO disclosed
WO-2012011125-A1 AGONISTS OF GPR40 CONNEXIOS LIFE SCIENCES PVT. LTD. (IN) 2012-01-26 WO disclosed
US-7276381-B2 Monomers and polymers having energy absorbing moieties of use in desorption/ionization of analytes BIO-RAD LABORATORIES, INC. (US) 2007-10-02 US disclosed
US-7276381-B2 Monomers and polymers having energy absorbing moieties of use in desorption/ionization of analytes BIO-RAD LABORATORIES, INC. (US) 2007-10-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130237571-A1 AGONISTS OF GPR40 GPR65, GPR55, GPR68 KDM4E 3722/4885ALDH1A1 2410/4885CISD1 3125/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.