SCHEMBL4377773

SCHEMBL4377773

CCc1cc2c(nc1-c1ccccc1)N=C(N)N(C)C2N

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
MAPT P10636 2/20 0.35
AKT1 P31749 1/20 0.32
AKT2 P31751 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
KDM4E B2RXH2 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
DHODH Q02127 1/20 0.31
BACE1 P56817 1/20 0.31
KDM5B Q9UGL1 1/20 0.30
HSD17B10 Q99714 1/20 0.30
ACHE P22303 1/20 0.30
TLR8 Q9NR97 1/20 0.30
DHFR P00374 1/20 0.30
HEXA P06865 1/20 0.30
HEXB P07686 1/20 0.30
PDE5A O76074 1/20 0.30
PTGDR2 Q9Y5Y4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4381715 0.87 ADK (0.41) BACE1TLR8DHFR
SCHEMBL4375812 0.81 ADORA1 (0.32) ADORA2AADORA1KDM4E
SCHEMBL3745220 0.73 PTPN1 (0.48) BACE1TLR8
SCHEMBL4511419 0.71 ALOX5AP (0.40) TLR8DHFR
SCHEMBL4528811 0.70 CTSD (0.44) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL3747039 0.68 ATP4A (0.32) BACE1
SCHEMBL3742648 0.64 PTPN1 (0.38)
SCHEMBL18825654 0.64 KDM4E (0.42) ALDH1A1MAPTADORA1KDM4EMEN1
SCHEMBL3734994 0.63 OPRM1 (0.35) BACE1
SCHEMBL3727477 0.62 PTPN1 (0.38) ALDH1A1ADORA2AADORA1BACE1TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910359-B1 PYRIDO [2 , 3-D]PYRIMIDINE-2 , 4-DIAMINE COMPOUNDS AS PTPlB INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-18 EP claimed