SCHEMBL4378501

SCHEMBL4378501

COc1ccc2c(c1)c(C(=O)C(=O)Nc1nc3ccccc3s1)c(C)n2Cc1ccc(Cl)cc1.COc1ccc2c(c1)c(C(=O)C(=O)Nc1nc3ccccc3s1)cn2Cc1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.47
PLA2G2A P14555 3/20 0.47
MAPT P10636 3/20 0.45
LMNA P02545 3/20 0.45
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 1/20 0.45
RGS12 O14924 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
PKM P14618 1/20 0.45
TSHR P16473 1/20 0.45
NFKB1 P19838 1/20 0.45
MAPK1 P28482 1/20 0.45
CYP2C19 P33261 1/20 0.45
GNAI1 P63096 1/20 0.45
PMP22 Q01453 1/20 0.45
KMT2A Q03164 1/20 0.45
HIF1A Q16665 1/20 0.45
CSNK1D P48730 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3011822 0.93 PLA2G2A (0.54) FAAHPLA2G2AMAPTLMNAALDH1A1
SCHEMBL3000071 0.92 CSNK1D (0.51) MAPTLMNAALDH1A1MEN1KMT2A
SCHEMBL4380867 0.81 PDE4A (0.56) FAAHPLA2G2AMAPTLMNAALDH1A1
SCHEMBL3004193 0.81 FAAH (0.56) FAAHPLA2G2AMAPTLMNAALDH1A1
SCHEMBL3001803 0.81 TUBB4A (0.47) PLA2G2AMAPTLMNAALDH1A1MEN1
SCHEMBL6086156 0.80 TUBB4A (0.63) MAPTLMNAALDH1A1MEN1CYP1A2
SCHEMBL4381471 0.79 FAAH (0.50) FAAHPLA2G2AMAPTLMNAALDH1A1
SCHEMBL4386750 0.78 FAAH (0.47) FAAHPLA2G2AMAPTLMNAALDH1A1
SCHEMBL4095457 0.77 FAAH (0.56) FAAHPLA2G2AMAPTLMNAALDH1A1
SCHEMBL4375897 0.77 FAAH (0.47) FAAHPLA2G2AMAPTLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed