Iodide

Iodide

SCHEMBL4379342

C[n+]1ccn(C(=O)N2CCC(c3cc(F)ccc3F)=CC2c2cccc(O)c2)c1.[I-]

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 19/20 0.54
KCNH2 Q12809 14/20 0.54
CASP3 P42574 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13624050 0.99 KIF11 (0.55) KIF11KCNH2CASP3
Iodide SCHEMBL5182650 0.83 KIF11 (0.65) KIF11KCNH2
SCHEMBL6532616 0.82 KIF11 (0.66) KIF11KCNH2
SCHEMBL4038431 0.82 KIF11 (0.66) KIF11KCNH2
SCHEMBL4374480 0.81 KIF11 (0.66) KIF11KCNH2CASP3
SCHEMBL13634117 0.76 KIF11 (0.82) KIF11KCNH2
SCHEMBL13624046 0.76 KIF11 (0.82) KIF11KCNH2
SCHEMBL4374455 0.72 KIF11 (0.79) KIF11KCNH2
SCHEMBL4059852 0.72 KIF11 (0.69) KIF11KCNH2
SCHEMBL14262984 0.71 KIF11 (0.68) KIF11KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622489-B2 Kinesin spindle protein inhibitor; antiproliferative agents; anticancer agents; 4-(2,5-difluorophenyl)-N-3-fluoropyrrolidin-3-yl)-2-hydroxymethyl-2-phenyl-2,5-dihydro-1N-pyrrol-1-carboxamide MERCK & CO., INC. (US) 2009-11-24 US disclosed
EP-1578724-A4 MITOTIC KINESIN INHIBITORS MERCK & CO INC (US) 2006-11-29 EP disclosed
US-20060052611-A1 Mitotic kinesin inhibitors MERCK SHARP & DOHME CORP. 2006-03-09 US disclosed
EP-1578724-A2 MITOTIC KINESIN INHIBITORS Merck & Co., Inc. (US) 2005-09-28 EP disclosed
WO-2004058700-A2 MITOTIC KINESIN INHIBITORS MERCK & CO., INC. (US) 2004-07-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060052611-A1 Mitotic kinesin inhibitors KIF5B, KIF2C, KIFC1 KIF11 10/4885KCNH2 1400/4885CASP3 3303/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.