SCHEMBL4381041

SCHEMBL4381041

COc1ncccc1C(=O)NC1(C)CCCCn2c1nc(-c1ccncc1)cc2=O

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
KDM4E B2RXH2 2/20 0.36
BRD4 O60885 1/20 0.35
BRPF1 P55201 1/20 0.35
GPR6 P46095 5/20 0.35
MAPT P10636 2/20 0.35
GAA P10253 1/20 0.35
TACR3 P29371 1/20 0.35
TSHR P16473 1/20 0.35
DHODH Q02127 1/20 0.34
GSK3B P49841 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
CYP2C9 P11712 1/20 0.34
GLA P06280 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ACKR3 P25106 1/20 0.34
ROCK2 O75116 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4384554 0.91 GSK3B (0.37) ALDH1A1KDM4EBRD4BRPF1GPR6
SCHEMBL4378591 0.88 GSK3B (0.38) BRD4BRPF1MAPTGAAGSK3B
SCHEMBL4387999 0.80 GSK3B (0.37) ALDH1A1TSHRGSK3BSMN1; SMN2
SCHEMBL4387224 0.80 ALDH1A1 (0.36) ALDH1A1KDM4EGPR6MAPTGAA
SCHEMBL4952879 0.78 MEN1 (0.47) ALDH1A1KDM4EGPR6KMT2AMEN1
SCHEMBL4383616 0.77 MEN1 (0.47) ALDH1A1BRD4BRPF1GPR6GAA
SCHEMBL2066100 0.77 GSK3B (0.43) ALDH1A1MAPTGSK3BKMT2AGLA
SCHEMBL4377844 0.75 MEN1 (0.45) BRD4BRPF1GPR6MAPTGAA
SCHEMBL4385699 0.73 GSK3B (0.35) GSK3B
SCHEMBL3373754 0.72 OPRD1 (0.41) GAAGSK3BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121635-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2009-11-25 EP claimed
WO-2008078196-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2008-07-03 WO claimed