SCHEMBL4382525

SCHEMBL4382525

O=C(O)C[C@@H](c1nc2ccccc2[nH]1)N1CCC(CCCC2=CC=C3CCCNC3N2)C1=O

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 7/20 0.46
ITGAV P06756 7/20 0.46
ITGA2B P08514 1/20 0.32
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KMT2A Q03164 1/20 0.31
FPR1 P21462 1/20 0.31
ATM Q13315 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
ITGA5 P08648 1/20 0.31
ITGB6 P18564 1/20 0.31
ITGB8 P26012 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4374458 0.86 ITGB3 (0.45) ITGB3ITGAVITGA2BLMNA
SCHEMBL4372884 0.85 ITGB3 (0.65) ITGB3ITGAVITGA2B
SCHEMBL4363508 0.85 ITGB3 (0.65) ITGB3ITGAVITGA2B
SCHEMBL4370537 0.85 ITGB3 (0.65) ITGB3ITGAVITGA2B
SCHEMBL7596620 0.85 ITGB8 (0.44) ITGB3ITGAVITGA2BKMT2AALDH1A1
SCHEMBL7594404 0.85 ITGB8 (0.44) ITGB3ITGAVITGA2BKMT2AALDH1A1
SCHEMBL7555650 0.85 ITGB8 (0.44) ITGB3ITGAVITGA2BKMT2AALDH1A1
SCHEMBL4368878 0.80 ITGAV (0.47) ITGB3ITGAVITGA2BITGA5ITGB6
SCHEMBL4386638 0.80 ITGB3 (0.43) ITGB3ITGAVITGA2BITGA5ITGB6
SCHEMBL4048448 0.80 ITGB3 (0.41) ITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047425-A4 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2009-04-22 EP disclosed
EP-1047425-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-11-02 EP disclosed
WO-1999030709-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed