SCHEMBL4383593

SCHEMBL4383593

CCOc1ccc2c(c1)c(C(=O)c1ncc(-c3ccccc3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1.COc1ccc2c(c1)c(C(=O)c1ncc(-c3ccccc3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1.O=C(c1cnc(-c2ccncn2)o1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2Cl)c2ccccc12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 8/20 0.33
ALOX5 P09917 4/20 0.33
EDNRB P24530 2/20 0.32
PLA2G2A P14555 2/20 0.32
F2RL3 Q96RI0 1/20 0.32
ACHE P22303 1/20 0.32
MEN1 O00255 1/20 0.31
RGS12 O14924 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
PKM P14618 1/20 0.31
TSHR P16473 1/20 0.31
NFKB1 P19838 1/20 0.31
MAPK1 P28482 1/20 0.31
CYP2C19 P33261 1/20 0.31
GNAI1 P63096 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2992472 0.95 ALOX5AP (0.32) ALOX5APALOX5
SCHEMBL2006472 0.88 ALOX5AP (0.36) ALOX5APALOX5F2RL3LMNAMAPT
SCHEMBL2006911 0.87 PLA2G2A (0.37) ALOX5APALOX5PLA2G2AF2RL3ACHE
SCHEMBL2002426 0.85 SLC26A4 (0.34) ALOX5APALOX5PLA2G2AF2RL3LMNA
SCHEMBL2006766 0.85 F2RL3 (0.40) ALOX5APEDNRBF2RL3ALDH1A1LMNA
SCHEMBL2010346 0.84 PLA2G2A (0.37) PLA2G2AF2RL3MEN1RGS12ALDH1A1
SCHEMBL2004514 0.84 F2RL3 (0.39) ALOX5APPLA2G2AF2RL3ALDH1A1CYP1A2
SCHEMBL2005424 0.84 ALOX5AP (0.42) ALOX5APALOX5CYP3A4CYP2C9
SCHEMBL1999823 0.83 F2RL3 (0.36) ALOX5APALOX5EDNRBF2RL3LMNA
SCHEMBL2009612 0.83 MEN1 (0.42) ALOX5APALOX5PLA2G2AACHEMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed