SCHEMBL2004514

SCHEMBL2004514

COc1ccc2c(c1)c(C(=O)c1ncc(-c3ccccc3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
F2RL3 Q96RI0 4/20 0.39
PLA2G2A P14555 7/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2D6 P10635 1/20 0.39
PTGS2 P35354 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
FAAH O00519 2/20 0.38
SLC26A4 O43511 1/20 0.37
POLB P06746 1/20 0.37
ALOX5AP P20292 2/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2008690 0.93 PLA2G2A (0.38) F2RL3PLA2G2ACYP1A2CYP3A4CYP2C9
SCHEMBL2006766 0.93 F2RL3 (0.40) F2RL3CYP1A2CYP3A4CYP2C9CYP2D6
SCHEMBL2001047 0.93 PLA2G2A (0.37) F2RL3PLA2G2ACYP1A2CYP3A4CYP2C9
SCHEMBL2006329 0.92 LMNA (0.38) CYP1A2CYP3A4CYP2C9CYP2D6MAPT
SCHEMBL2004225 0.91 PLA2G2A (0.45) PLA2G2ACYP1A2CYP3A4CYP2C9PTGS2
SCHEMBL2000385 0.91 FAAH (0.38) F2RL3PLA2G2AFAAH
SCHEMBL2005400 0.90 PPARG (0.36) CYP1A2CYP3A4CYP2C9CYP2D6MAPT
SCHEMBL2006669 0.90 PLA2G2A (0.41) F2RL3PLA2G2ACYP1A2CYP3A4CYP2C9
SCHEMBL2002966 0.89 L3MBTL1 (0.40) CYP1A2CYP3A4CYP2C9CYP2D6MAPT
SCHEMBL2008823 0.89 LMNA (0.41) CYP1A2CYP3A4CYP2C9CYP2D6TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed