SCHEMBL4385085

SCHEMBL4385085

[CH2]CNc1nc(NCc2ccc(F)c(Cl)c2)ncc1[N+](=O)[O-]

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCQ Q04759 18/20 0.54
HDAC3 O15379 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
STK17A Q9UEE5 1/20 0.47
DCLK1 O15075 1/20 0.45
MAP4K4 O95819 1/20 0.45
CDK1 P06493 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
PIM1 P11309 1/20 0.45
CYP2C9 P11712 1/20 0.45
PRKACA P17612 1/20 0.45
CDK2 P24941 1/20 0.45
MATK P42679 1/20 0.45
FRK P42685 1/20 0.45
CSNK1D P48730 1/20 0.45
CLK2 P49760 1/20 0.45
GSK3A P49840 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4389712 0.91 PRKCQ (0.54) PRKCQSTK17ADCLK1MAP4K4CDK1
SCHEMBL4384306 0.90 PRKCQ (0.53) PRKCQSTK17A
SCHEMBL4387931 0.86 PRKCQ (0.67) PRKCQSTK17ADCLK1MAP4K4CDK1
SCHEMBL4387612 0.85 PRKCQ (0.68) PRKCQHDAC3HDAC1HDAC2HDAC6
SCHEMBL4379701 0.85 MAPT (0.46) PRKCQHDAC3HDAC1HDAC2HDAC6
SCHEMBL3179956 0.84 PRKCQ (0.49) PRKCQHDAC3HDAC1HDAC2HDAC6
SCHEMBL4392873 0.84 PRKCQ (0.67) PRKCQCYP3A4CYP2C9
SCHEMBL13671819 0.83 PRKCQ (0.68) PRKCQDCLK1MAP4K4CDK1CYP3A4
SCHEMBL4380044 0.82 PRKCQ (0.69) PRKCQ
SCHEMBL4386385 0.81 HDAC3 (0.51) HDAC3HDAC1HDAC2HDAC6STK17A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2131844-A1 PTERIDINONE DERIVATIVES FOR USE AS STEAROYL CoA DESATURASE INHIBITORS CV Therapeutics Inc. (US) 2009-12-16 EP disclosed
WO-2008123891-A1 PTERIDINONE DERIVATIVES FOR USE AS STEAROYL CoA DESATURASE INHIBITORS CV THERAPEUTICS, INC. (US) 2008-10-16 WO disclosed