SCHEMBL4389712

SCHEMBL4389712

[CH2]CNc1nc(NCc2ccc(Cl)c(F)c2)ncc1[N+](=O)[O-]

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCQ Q04759 19/20 0.54
CYP3A4 P08684 2/20 0.45
CYP2C9 P11712 2/20 0.45
DCLK1 O15075 1/20 0.45
MAP4K4 O95819 1/20 0.45
CDK1 P06493 1/20 0.45
CYP2D6 P10635 1/20 0.45
PIM1 P11309 1/20 0.45
PRKACA P17612 1/20 0.45
CDK2 P24941 1/20 0.45
MATK P42679 1/20 0.45
FRK P42685 1/20 0.45
CSNK1D P48730 1/20 0.45
CLK2 P49760 1/20 0.45
GSK3A P49840 1/20 0.45
GSK3B P49841 1/20 0.45
IRAK1 P51617 1/20 0.45
RPS6KA3 P51812 1/20 0.45
CDK5 Q00535 1/20 0.45
PRKCD Q05655 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4385085 0.91 PRKCQ (0.54) PRKCQCYP3A4CYP2C9DCLK1MAP4K4
SCHEMBL4384306 0.90 PRKCQ (0.53) PRKCQSTK17A
SCHEMBL3182009 0.84 PRKCQ (0.49) PRKCQCYP3A4CYP2C9STK17A
SCHEMBL4392873 0.84 PRKCQ (0.67) PRKCQCYP3A4CYP2C9
SCHEMBL4387931 0.84 PRKCQ (0.67) PRKCQCYP3A4CYP2C9DCLK1MAP4K4
SCHEMBL4387612 0.83 PRKCQ (0.68) PRKCQCYP3A4CYP2C9DCLK1MAP4K4
SCHEMBL4380044 0.82 PRKCQ (0.69) PRKCQ
SCHEMBL4387694 0.81 DYRK1A (0.41) PRKCQDYRK1ASTK17A
SCHEMBL4384358 0.79 PRKCQ (0.65) PRKCQGSK3B
SCHEMBL3179956 0.76 PRKCQ (0.49) PRKCQCYP3A4CYP2C9STK17A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2131844-A1 PTERIDINONE DERIVATIVES FOR USE AS STEAROYL CoA DESATURASE INHIBITORS CV Therapeutics Inc. (US) 2009-12-16 EP disclosed
WO-2008123891-A1 PTERIDINONE DERIVATIVES FOR USE AS STEAROYL CoA DESATURASE INHIBITORS CV THERAPEUTICS, INC. (US) 2008-10-16 WO disclosed