SCHEMBL4387727

SCHEMBL4387727

Cc1ccnc(C=O)c1N

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 6/20 0.54
NOS3 P29474 5/20 0.54
LMNA P02545 2/20 0.37
LIMK1 P53667 1/20 0.37
CCR1 P32246 2/20 0.35
CCR5 P51681 2/20 0.35
CCR8 P51685 2/20 0.35
NOS1 P29475 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PSMD14 O00487 1/20 0.32
COPS5 Q92905 1/20 0.32
POLB P06746 1/20 0.32
CD44 P16070 1/20 0.32
ALDH1A1 P00352 3/20 0.31
TSHR P16473 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21899450 0.79 NOS2 (0.54) NOS2NOS3LMNALIMK1CCR1
SCHEMBL2085241 0.78 NOS2 (0.46) NOS2NOS3LMNACCR1CCR5
SCHEMBL25346137 0.75 CCR1 (0.32) NOS2NOS3CCR1CCR5CCR8
SCHEMBL8688305 0.75 KDM4C (0.39) NOS2NOS3LMNACCR1CCR5
SCHEMBL20767182 0.75 CCR1 (0.35) NOS2NOS3LMNACCR1CCR5
SCHEMBL12468608 0.75 CCR1 (0.35) NOS2NOS3LMNACCR1CCR5
SCHEMBL3716910 0.75 CCR1 (0.35) NOS2NOS3LMNACCR1CCR5
SCHEMBL20135919 0.75 NOS2 (0.35) NOS2NOS3LMNALIMK1CCR1
SCHEMBL28272737 0.72 MAOA (0.37) NOS2NOS3LIMK1CCR1CCR5
SCHEMBL1223407 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090298891-A1 Methods of Treating or Preventing Cancer Using Pyridine Carboxaldehyde Pyridine Thiosemicarbazone Radiosensitizing Agents GOVERNMENT OF THE US, AS REPRESENTED BY THE SECRETADY OF HEALTH AND HUMAN SERVICES (US) 2009-12-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090298891-A1 Methods of Treating or Preventing Cancer Using Pyridine Carboxaldehyde Pyridine Thiosemicarbazone Radiosensitizing Agents DPYD, NTPCR, RRM2B NOS2 1357/4885NOS3 1356/4885LMNA 3037/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.