SCHEMBL20135919

SCHEMBL20135919

Cc1ccnc(C=O)c1-c1ncccn1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 5/20 0.35
NOS3 P29474 4/20 0.35
NOS1 P29475 1/20 0.35
CCR1 P32246 3/20 0.33
CCR8 P51685 3/20 0.33
CCR5 P51681 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 2/20 0.32
TRIM24 O15164 1/20 0.32
TRIM33 Q9UPN9 1/20 0.32
TSHR P16473 1/20 0.32
CYP2A6 P11509 1/20 0.32
LIMK1 P53667 1/20 0.31
HTR2B P41595 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C19 P33261 1/20 0.30
PLAU P00749 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4387727 0.75 NOS2 (0.54) NOS2NOS3NOS1CCR1CCR8
SCHEMBL20135885 0.74 ALDH1A1 (0.50) NOS2NOS3NOS1CCR1CCR8
SCHEMBL570133 0.74
SCHEMBL2085241 0.74 NOS2 (0.46) NOS2NOS3CCR1CCR8CCR5
SCHEMBL29426573 0.74
SCHEMBL3340081 0.73 NOS3 (0.42) NOS2NOS3NOS1CCR1CCR8
SCHEMBL8688305 0.71 KDM4C (0.39) NOS2NOS3CCR1CCR8CCR5
SCHEMBL3716910 0.71 CCR1 (0.35) NOS2NOS3CCR1CCR8CCR5
SCHEMBL20767182 0.71 CCR1 (0.35) NOS2NOS3CCR1CCR8CCR5
SCHEMBL12468608 0.71 CCR1 (0.35) NOS2NOS3CCR1CCR8CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP claimed