SCHEMBL4391765

SCHEMBL4391765

C#Cc1cc(Cl)cc(C#N)c1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 7/20 0.37
VCAM1 P19320 1/20 0.36
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
TTR P02766 2/20 0.33
ALB P02768 2/20 0.33
CYP1A2 P05177 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
KCNH2 Q12809 1/20 0.33
GPR35 Q9HC97 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19267579 0.87 TTR (0.40) VCAM1TTRALBMEN1KMT2A
SCHEMBL5852713 0.87 VCAM1 (0.43) GRM5VCAM1MAOAMAOBTTR
SCHEMBL718951 0.82 TSHR (0.50)
SCHEMBL633226 0.82 TSHR (0.50) GRM5VCAM1MAOAMAOBTTR
SCHEMBL2767750 0.76 GRM5 (0.41) GRM5
SCHEMBL16958396 0.76 GRM5 (0.37) GRM5VCAM1MAOAMAOBTTR
SCHEMBL16954469 0.76 GRM5 (0.37) GRM5VCAM1MAOAMAOBTTR
SCHEMBL18934332 0.76 ALDH1A1 (0.42) GRM5VCAM1TTRALBMEN1
SCHEMBL26002403 0.73 TTR (0.35) TTRALBMEN1KMT2A
Cyanide SCHEMBL11880265 0.73 TTR (0.46) GRM5VCAM1TTRALBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8383658-B2 Isoxazole based neuronal nicotinic receptor ligands and methods of use ABBOTT LABORATORIES (US) 2013-02-26 US disclosed
US-20090306096-A1 Novel Isoxazoles and Methods of Use Thereof ABBOTT LABORATORIES (US) 2009-12-10 US disclosed
WO-2009149135-A1 BIS (HETERO ) ARYL SUBSTITUTED ISOXAZOLES FOR USE AS NEURONAL NICOTINIC RECEPTOR MODULATORS ABBOTT LABORATORIES (US) 2009-12-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090306096-A1 Novel Isoxazoles and Methods of Use Thereof XDH, PRDX5, CYP4X1 GRM5 1012/4885VCAM1 2739/4885MAOA 508/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.