SCHEMBL4396565

SCHEMBL4396565

COc1ccc(CCN(CC(N)=O)C(=O)C2CC(=O)N(CCc3ccc(Cl)cc3Cl)CC(=O)N2CCC(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APAF1 O14727 6/20 0.83
CASP3 P42574 6/20 0.83
CASP9 P55211 6/20 0.83
CYCS P99999 6/20 0.83
ACHE P22303 1/20 0.40
CCR5 P51681 2/20 0.37
C5AR1 P21730 1/20 0.36
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CTSD P07339 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4401180 0.94 APAF1 (0.91) APAF1CASP3CASP9CYCSACHE
SCHEMBL4391634 0.91 APAF1 (0.86) APAF1CASP3CASP9CYCSACHE
SCHEMBL4388693 0.91 APAF1 (1.00) APAF1CASP3CASP9CYCSACHE
SCHEMBL4541497 0.90 APAF1 (0.86) APAF1CASP3CASP9CYCSACHE
SCHEMBL12009680 0.88 APAF1 (0.63) APAF1CASP3CASP9CYCSACHE
SCHEMBL4395653 0.88 APAF1 (0.90) APAF1CASP3CASP9CYCSACHE
SCHEMBL4398368 0.88 APAF1 (0.87) APAF1CASP3CASP9CYCSACHE
SCHEMBL4397286 0.86 APAF1 (0.90) APAF1CASP3CASP9CYCSACHE
SCHEMBL13875429 0.84 APAF1 (0.58) APAF1CASP3CASP9CYCSACHE
SCHEMBL4391987 0.82 APAF1 (0.77) APAF1CASP3CASP9CYCSACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963357-B1 COMPOUNDS FOR THE INHIBITION OF APOPTOSIS SALVAT LAB SA (ES) 2009-12-09 EP disclosed