SCHEMBL4396601

SCHEMBL4396601

C[C@H]1CN([C@@H](C)CN2CCC(NC(=O)Oc3cc4c(OCC5CCC5)cccc4[nH]3)CC2)C[C@H](O)[C@@H]1O

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GUCY1B2 O75343 1/20 0.34
GUCY1A2 P33402 1/20 0.34
GUCY1A1 Q02108 1/20 0.34
GUCY1B1 Q02153 1/20 0.34
PARP1 P09874 2/20 0.33
SLC6A4 P31645 3/20 0.32
DRD2 P14416 2/20 0.32
HTR2B P41595 1/20 0.32
HTR1A P08908 6/20 0.32
LMNA P02545 1/20 0.32
ACACB O00763 1/20 0.32
KMT2A Q03164 1/20 0.32
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
ADRB3 P13945 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4396942 0.92 PARP1 (0.34) GUCY1B2GUCY1A2GUCY1A1GUCY1B1PARP1
SCHEMBL4405858 0.92 PARP1 (0.34) GUCY1B2GUCY1A2GUCY1A1GUCY1B1PARP1
SCHEMBL914354 0.89 KMT2A (0.40) GUCY1B2GUCY1A2GUCY1A1GUCY1B1PARP1
SCHEMBL4396432 0.89 HTR1A (0.36) PARP1SLC6A4HTR1ALMNAKMT2A
SCHEMBL4551076 0.87 HTR1A (0.33) GUCY1B2GUCY1A2GUCY1A1GUCY1B1PARP1
SCHEMBL4403759 0.85 HTR1A (0.37) PARP1SLC6A4DRD2HTR2BHTR1A
SCHEMBL4397029 0.84 DRD2 (0.33) SLC6A4DRD2HTR1AADRB3
SCHEMBL4398650 0.83 GUCY1B2 (0.35) GUCY1B2GUCY1A2GUCY1A1GUCY1B1PARP1
SCHEMBL4400739 0.81 GUCY1B2 (0.37) GUCY1B2GUCY1A2GUCY1A1GUCY1B1PARP1
SCHEMBL913924 0.81 KMT2A (0.42) GUCY1B2GUCY1A2GUCY1A1GUCY1B1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed