SCHEMBL4551076

SCHEMBL4551076

C[C@H]1CN([C@@H](CO)CN2CCC(NC(=O)Oc3cc4c(OCC5CCC5)cccc4[nH]3)CC2)CC[C@@H]1O

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.33
SLC6A4 P31645 1/20 0.32
PARP1 P09874 2/20 0.32
GUCY1B2 O75343 1/20 0.31
GUCY1A2 P33402 1/20 0.31
GUCY1A1 Q02108 1/20 0.31
GUCY1B1 Q02153 1/20 0.31
LMNA P02545 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4405858 0.92 PARP1 (0.34) HTR1ASLC6A4PARP1GUCY1B2GUCY1A2
SCHEMBL4396942 0.92 PARP1 (0.34) HTR1ASLC6A4PARP1GUCY1B2GUCY1A2
SCHEMBL914741 0.89 KMT2A (0.38) HTR1APARP1GUCY1B2GUCY1A2GUCY1A1
SCHEMBL4398650 0.87 GUCY1B2 (0.35) HTR1ASLC6A4PARP1GUCY1B2GUCY1A2
SCHEMBL4396601 0.87 GUCY1B2 (0.34) HTR1ASLC6A4PARP1GUCY1B2GUCY1A2
SCHEMBL4396432 0.84 HTR1A (0.36) HTR1ASLC6A4PARP1LMNAKMT2A
SCHEMBL2321353 0.81 GUCY1B2 (0.31) GUCY1B2GUCY1A2GUCY1A1GUCY1B1KMT2A
SCHEMBL4403759 0.81 HTR1A (0.37) HTR1ASLC6A4PARP1LMNA
SCHEMBL913924 0.80 KMT2A (0.42) PARP1GUCY1B2GUCY1A2GUCY1A1GUCY1B1
SCHEMBL914364 0.80 KMT2A (0.42) PARP1GUCY1B2GUCY1A2GUCY1A1GUCY1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed