SCHEMBL4396633

SCHEMBL4396633

C[C@H]1CN([C@@H](C)CN2CCC(NC(=O)Oc3cc4c(OCc5coc6ccc(F)cc56)cccc4[nH]3)CC2)CC[C@@H]1O

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.34
HTR1A P08908 5/20 0.33
MCHR1 Q99705 10/20 0.32
KCNH2 Q12809 8/20 0.32
MCHR2 Q969V1 4/20 0.32
ADRB2 P07550 1/20 0.31
ADRB1 P08588 1/20 0.31
ADRB3 P13945 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
WNT1 P04628 1/20 0.31
DYRK1A Q13627 1/20 0.31
SLC6A4 P31645 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4409298 0.95 MCHR1 (0.35) HTR1AMCHR1KCNH2MCHR2
SCHEMBL4404719 0.95 SOS1 (0.34) SOS1HTR1AMCHR1KCNH2MCHR2
SCHEMBL4396436 0.93 DRD2 (0.33) HTR1AADRB2ADRB1ADRB3MAOA
Hydrochloric Acid SCHEMBL4541892 0.93 SOS1 (0.33) SOS1HTR1AMCHR1MAOAMAOB
Hydrochloric Acid SCHEMBL4412704 0.92 HTR1A (0.31) HTR1ASLC6A4
Hydrochloric Acid SCHEMBL4396450 0.91 SOS1 (0.36) SOS1HTR1AMCHR1KCNH2MCHR2
Hydrochloric Acid SCHEMBL4399336 0.91 HTR1A (0.33) HTR1AMCHR1KCNH2MCHR2ADRB2
SCHEMBL914253 0.90 KMT2A (0.36) SOS1MCHR1KCNH2MCHR2WNT1
SCHEMBL4398647 0.90 KDM4E (0.33) HTR1AMCHR1ADRB2ADRB1ADRB3
SCHEMBL4404545 0.89 MAOB (0.39) MCHR1KCNH2ADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed