SCHEMBL4397065

SCHEMBL4397065

COCCN(C)S(=O)(=O)c1ccc(C(=N)NO)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.46
NPSR1 Q6W5P4 2/20 0.44
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 4/20 0.42
TSHR P16473 3/20 0.42
LMNA P02545 2/20 0.42
RXFP1 Q9HBX9 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CA12 O43570 2/20 0.41
CA9 Q16790 2/20 0.41
CA1 P00915 1/20 0.41
HTT P42858 1/20 0.40
MMP1 P03956 1/20 0.40
MMP9 P14780 1/20 0.40
MMP13 P45452 1/20 0.40
ADAM17 P78536 1/20 0.40
RECQL P46063 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17290956 0.80 KMT2A (0.51) CASP3NPSR1ALDH1A1KDM4ETSHR
SCHEMBL3054683 0.80 CA12 (0.55) CASP3ALDH1A1KDM4ELMNARXFP1
SCHEMBL17290492 0.78 CASP3 (0.46) CASP3NPSR1ALDH1A1KDM4ETSHR
SCHEMBL3917930 0.78 SIGMAR1 (0.55) CASP3ALDH1A1KDM4ETSHRLMNA
SCHEMBL4394070 0.78 MAPT (0.48) NPSR1ALDH1A1KDM4ETSHRLMNA
SCHEMBL10090152 0.76 CASP3 (0.58) CASP3ALDH1A1LMNACA12CA9
SCHEMBL4768851 0.75 CASP3 (0.53) CASP3ALDH1A1TSHRLMNACYP3A4
SCHEMBL6103289 0.75 SIGMAR1 (0.55) CASP3ALDH1A1LMNAHTTMMP13
SCHEMBL4394101 0.75 HTT (0.58) NPSR1ALDH1A1TSHRLMNACA12
SCHEMBL19001342 0.75 MAPK1 (0.55) CASP3ALDH1A1LMNAHTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed