SCHEMBL4397673

SCHEMBL4397673

CN(CCCCc1ccccc1Sc1c[nH]c2ccccc12)C(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.44
NPC1 O15118 1/20 0.44
CDK4 P11802 8/20 0.41
CCND1 P24385 8/20 0.41
SLC6A4 P31645 1/20 0.40
POLB P06746 1/20 0.40
GFER P55789 1/20 0.39
HTR1A P08908 1/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
MAOA P21397 1/20 0.38
ADRA1D P25100 1/20 0.38
HTR1B P28222 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
HTR7 P34969 1/20 0.38
ADRA1A P35348 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4391454 0.97 SMN1; SMN2 (0.45) SMN1; SMN2NPC1CDK4CCND1SLC6A4
SCHEMBL4387834 0.93 CDK4 (0.47) CDK4CCND1
SCHEMBL4394022 0.87 NPC1 (0.38) SMN1; SMN2NPC1CDK4CCND1SLC6A4
SCHEMBL4389267 0.87 CDK4 (0.39) SMN1; SMN2NPC1CDK4CCND1SLC6A4
SCHEMBL4396116 0.86 SLC6A4 (0.43) SMN1; SMN2NPC1CDK4CCND1SLC6A4
SCHEMBL4393850 0.86 ACHE (0.40) SMN1; SMN2NPC1CDK4CCND1SLC6A4
SCHEMBL4963737 0.84 TACR1 (0.40) CDK4CCND1HTR1ANAMPT
SCHEMBL4388059 0.84 PTGS2 (0.34) SMN1; SMN2NPC1CDK4CCND1SLC6A4
SCHEMBL4388601 0.83 SLC6A4 (0.47) SMN1; SMN2NPC1CDK4CCND1SLC6A4
SCHEMBL4386318 0.83 CDK4 (0.48) CDK4CCND1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893575-B1 2-(1H-INDOLYLSULFANYL)-ARYL AMINE DERIVATIVES H LUNDBECK AS (DK) 2017-01-11 EP disclosed
US-7629473-B2 2-(1H-indolylsulfanyl)-aryl amine derivatives H. LUNDBECK A/S (DK) 2009-12-08 US disclosed
US-20060287382-A1 2-(1H-indolylsulfanyl)-aryl amine derivatives H. LUNDBECK A/S (DK) 2006-12-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060287382-A1 2-(1H-indolylsulfanyl)-aryl amine derivatives CYP11B2, CYP1A2, CYP4B1 SMN1; SMN2 907/4885NPC1 442/4885CDK4 550/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.