SCHEMBL4398942

SCHEMBL4398942

OCc1ccc[n+](CCOCCOCCOCC[n+]2cccc(CO)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BCHE P06276 3/20 0.47
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
KDM4E B2RXH2 2/20 0.37
ACHE P22303 2/20 0.37
GGPS1 O95749 1/20 0.36
TSHR P16473 1/20 0.35
HDAC1 Q13547 2/20 0.35
CYP2D6 P10635 1/20 0.35
HDAC4 P56524 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2175968 0.98 BCHE (0.46) BCHEGRIN1GRIN2AKDM4EACHE
SCHEMBL4399006 0.83 GGPS1 (0.44) BCHEGRIN1GRIN2AKDM4EGGPS1
Hydrochloric Acid SCHEMBL2177623 0.82 HDAC1 (0.46) BCHEGRIN1GRIN2AKDM4EGGPS1
SCHEMBL21490429 0.81 TSHR (0.44) KDM4ETSHRHDAC1CYP2D6HDAC4
Bromide SCHEMBL20544414 0.79 KDM4E (0.58) BCHEKDM4EACHEHDAC1HDAC4
SCHEMBL28051020 0.76 GGPS1 (0.34) KDM4EGGPS1CYP2D6
SCHEMBL294104 0.75 LMNA (0.44) KDM4EACHE
Bromide SCHEMBL7696012 0.75 CYP2D6 (0.55) BCHEKDM4EACHETSHRHDAC1
SCHEMBL4401483 0.74 BCHE (0.50) BCHEGRIN1GRIN2AKDM4EACHE
SCHEMBL295339 0.73 TSHR (0.41) KDM4EGGPS1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178678-B2 Bis-quaternary ammonium salts and methods for modulating neuronal nicotinic acetylcholine receptors UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2012-05-15 US disclosed
US-20100069432-A1 Bis-Quaternary Ammonium Salts and Methods for Modulating Neuronal Nicotinic Acetylcholine Receptors UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2010-03-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100069432-A1 Bis-Quaternary Ammonium Salts and Methods for Modulating Neuronal Nicotinic Acetylcholine Receptors CHRNA2, CHRNA5, CHRNA4 BCHE 39/4885GRIN1 29/4885GRIN2A 33/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.