SCHEMBL440348

SCHEMBL440348

Nc1c(Br)cnc2ccc(OC(F)(F)F)cc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
TP53 P04637 2/20 0.44
GMNN O75496 1/20 0.44
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
GAA P10253 1/20 0.44
CYP2C9 P11712 1/20 0.44
PKM P14618 1/20 0.44
ALOX15 P16050 1/20 0.44
NFKB1 P19838 1/20 0.44
SLC6A2 P23975 1/20 0.44
SCN4A P35499 1/20 0.44
BLM P54132 1/20 0.44
PMP22 Q01453 1/20 0.44
SLC6A3 Q01959 1/20 0.44
PDE4D Q08499 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL439912 0.88 ALOX5AP (0.42) NPC1RAB9ATP53GMNNUSP2
SCHEMBL437175 0.82 NPC1 (0.44) NPC1RAB9ATP53GMNNUSP2
SCHEMBL439635 0.80 APP (0.48) LMNACYP1A2CYP3A4MAPK1ABCC8
SCHEMBL439021 0.78 KMT2A (0.55) NPC1TP53LMNACYP1A2CYP3A4
SCHEMBL436530 0.77 BACE1 (0.42) SCN4AALOX5APFEN1KDRKDM4E
SCHEMBL439853 0.74 BCHE (0.43) LMNADHODHACHE
SCHEMBL438613 0.74 BCHE (0.45) LMNASMN1; SMN2ACHE
SCHEMBL4271192 0.74 NR4A2 (0.51) NPC1RAB9ATP53GMNNUSP2
SCHEMBL30513837 0.74 MAP4K4 (0.54) NPC1RAB9ATP53GMNNUSP2
SCHEMBL22589620 0.72 DDR1 (0.44) NPC1RAB9ATP53GMNNUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed