SCHEMBL439853

SCHEMBL439853

Nc1c(Br)cnc2ccc(F)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 5/20 0.43
ACHE P22303 5/20 0.43
GRIN1 Q05586 5/20 0.43
GRIN2A Q12879 5/20 0.43
PARP1 P09874 1/20 0.41
MAP4K4 O95819 2/20 0.39
BACE1 P56817 1/20 0.38
AXL P30530 1/20 0.36
GFER P55789 1/20 0.36
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
USP10 Q14694 1/20 0.36
PIK3C3 Q8NEB9 1/20 0.36
USP13 Q92995 1/20 0.36
TYMS P04818 1/20 0.36
DHODH Q02127 1/20 0.35
LMNA P02545 1/20 0.35
PIK3CD O00329 1/20 0.35
PIK3CA P42336 1/20 0.35
MTOR P42345 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL439004 0.86 ACHE (0.43) ACHEMAP4K4BACE1
SCHEMBL438613 0.81 BCHE (0.45) BCHEACHEGRIN1GRIN2ABACE1
SCHEMBL10385174 0.81 BCHE (0.45) BCHEACHEGRIN1GRIN2APARP1
SCHEMBL437551 0.79 NR4A2 (0.51) BCHEACHEGRIN1GRIN2APARP1
SCHEMBL442244 0.79 ACHE (0.43) BCHEACHEGRIN1GRIN2APARP1
SCHEMBL20494939 0.79 PARP1 (0.41) BCHEACHEGRIN1GRIN2APARP1
SCHEMBL439645 0.79 ACHE (0.46) BCHEACHEGRIN1GRIN2APARP1
SCHEMBL29391085 0.79 PARP1 (0.41) BCHEACHEGRIN1GRIN2APARP1
SCHEMBL436530 0.78 BACE1 (0.42) MAP4K4BACE1AXLCCNCCDK8
SCHEMBL439366 0.75 ALDH1A1 (0.46) TYMSLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed