SCHEMBL4404902

SCHEMBL4404902

CC(=O)c1ccc2[nH]n(C)c(=O)c2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.51
KIF11 P52732 1/20 0.45
HTR1A P08908 1/20 0.42
HTR1D P28221 1/20 0.42
HTR1B P28222 1/20 0.42
SLC2A1 P11166 1/20 0.42
ACACB O00763 1/20 0.41
ACACA Q13085 1/20 0.41
KDM4E B2RXH2 1/20 0.40
TP53 P04637 1/20 0.40
HRH4 Q9H3N8 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
ERCC1 P07992 1/20 0.38
DNASE1 P24855 1/20 0.38
FEN1 P39748 1/20 0.38
ERCC4 Q92889 1/20 0.38
PARP1 P09874 1/20 0.38
KMT2A Q03164 1/20 0.38
NR1H2 P55055 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2671424 0.87 ALOX5 (0.51) ALOX5KIF11ACACBACACAKDM4E
SCHEMBL4402967 0.87 ALOX5 (0.51) ALOX5KIF11SLC2A1ACACBACACA
SCHEMBL4400592 0.83 ALOX5 (0.47) ALOX5KIF11ACACBACACAKDM4E
SCHEMBL2671133 0.73 KDM4E (0.52) ALOX5KDM4EPARP1KMT2AALDH1A1
SCHEMBL30366673 0.72 KIF11 (0.74) KIF11HTR1AHTR1DHTR1BSLC2A1
SCHEMBL31506909 0.72 KIF11 (0.74) KIF11HTR1AHTR1DHTR1BSLC2A1
SCHEMBL2333579 0.72 KIF11 (0.74) KIF11HTR1AHTR1DHTR1BSLC2A1
SCHEMBL2056375 0.71 ALOX5 (0.53) ALOX5KIF11HTR1AHTR1DHTR1B
SCHEMBL2054602 0.71 ALOX5 (0.53) ALOX5KIF11HTR1AHTR1DHTR1B
SCHEMBL21156818 0.70 LMNA (0.51) KIF11HRH4KMT2ANR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012056372-A1 N1/N2-LACTAM ACETYL-CoA CARBOXYLASE INHIBITORS PFIZER INC. (US) 2012-05-03 WO disclosed