SCHEMBL4404909

SCHEMBL4404909

COc1cccc2ncc(C(C)=O)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 2/20 0.46
ALDH1A1 P00352 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.44
HSD17B10 Q99714 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
EGFR P00533 1/20 0.44
ERBB2 P04626 1/20 0.44
HPGDS O60760 1/20 0.44
PDE10A Q9Y233 1/20 0.44
MAP4K4 O95819 1/20 0.43
CSNK1G2 P78368 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43
MAP4K5 Q9Y4K4 1/20 0.43
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
MGLL Q99685 1/20 0.42
ACACB O00763 1/20 0.42
ACACA Q13085 1/20 0.42
PDE3B Q13370 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30829596 0.88 MGAM (0.51) ALDH1A1SMN1; SMN2HSD17B10L3MBTL1HPGDS
SCHEMBL30440820 0.88 MGAM (0.51) ALDH1A1SMN1; SMN2HSD17B10L3MBTL1HPGDS
SCHEMBL2202272 0.88 MGAM (0.51) ALDH1A1SMN1; SMN2HSD17B10L3MBTL1HPGDS
SCHEMBL19329127 0.87 HPGDS (0.52) SMN1; SMN2HSD17B10L3MBTL1EGFRERBB2
SCHEMBL2201313 0.87 ALPL (0.47) ALDH1A1SMN1; SMN2HSD17B10L3MBTL1HPGDS
SCHEMBL4137438 0.84 ACACB (0.44) ALDH1A1SMN1; SMN2HSD17B10L3MBTL1HPGDS
SCHEMBL2199970 0.82 PDGFRB (0.52) RXFP1ALDH1A1SMN1; SMN2LMNAMEN1
SCHEMBL27909233 0.79 ALDH1A1 (0.56) ALDH1A1PDE10AMTNR1AMTNR1BLMNA
SCHEMBL26317945 0.78 SLC2A1 (0.51) RXFP1ALDH1A1SMN1; SMN2SRCTGFBR1
SCHEMBL11152987 0.77 MGAM (0.45) ALDH1A1SMN1; SMN2MAP4K4CSNK1G2CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012056372-A1 N1/N2-LACTAM ACETYL-CoA CARBOXYLASE INHIBITORS PFIZER INC. (US) 2012-05-03 WO disclosed