SCHEMBL4405432

SCHEMBL4405432

C[C@@H](CN1CCC(NC(=O)Oc2cc3c(OCc4coc5cccc(Cl)c45)cccc3[nH]2)CC1)N1CCC(O)CC1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.35
HTR1A P08908 7/20 0.32
SLC6A4 P31645 1/20 0.32
HTR7 P34969 1/20 0.31
ACHE P22303 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
ADRB2 P07550 1/20 0.31
ADRB1 P08588 1/20 0.31
ADRB3 P13945 1/20 0.31
CCR5 P51681 1/20 0.31
TLR9 Q9NR96 1/20 0.31
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4401792 0.91 DRD2 (0.35) HTR1ASLC6A4ACHEMAOAMAOB
Hydrochloric Acid SCHEMBL4403798 0.90 MAOB (0.33) MCHR1HTR1AHTR7MAOAMAOB
SCHEMBL913655 0.90 MCHR1 (0.39) MCHR1HTR7ACHEMAOAMAOB
Hydrochloric Acid SCHEMBL4396448 0.89 SOS1 (0.33) MCHR1HTR1ASLC6A4HTR7MAOB
Hydrochloric Acid SCHEMBL4409021 0.89 SOS1 (0.36) MCHR1HTR1ASLC6A4HTR7MAOA
SCHEMBL4400742 0.89 MCHR1 (0.36) MCHR1HTR1ASLC6A4ACHEMAOB
Hydrochloric Acid SCHEMBL4405309 0.88 HTR1A (0.36) MCHR1HTR1ASLC6A4ADRB2ADRB1
Hydrochloric Acid SCHEMBL4396591 0.88 HTR1A (0.34) MCHR1HTR1ASLC6A4TLR9TLR8
Hydrochloric Acid SCHEMBL4396450 0.87 SOS1 (0.36) MCHR1HTR1ASLC6A4MAOAMAOB
Hydrochloric Acid SCHEMBL4403801 0.87 HTR1A (0.37) MCHR1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed