SCHEMBL4400742

SCHEMBL4400742

COc1cc(OC)c2c(COc3cccc4[nH]c(OC(=O)NC5CCN(C[C@H](C)N6CCC(O)CC6)CC5)cc34)coc2c1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 4/20 0.36
MAOB P27338 2/20 0.35
ADRB2 P07550 3/20 0.34
ADRB1 P08588 3/20 0.34
ADRB3 P13945 3/20 0.34
HTR1A P08908 2/20 0.34
SLC6A4 P31645 1/20 0.34
SLC2A1 P11166 1/20 0.33
KCNH2 Q12809 2/20 0.32
TLR9 Q9NR96 1/20 0.32
TLR8 Q9NR97 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
MAPT P10636 1/20 0.32
ACHE P22303 3/20 0.32
BCHE P06276 1/20 0.32
SIGMAR1 Q99720 1/20 0.31
USP2 O75604 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4400748 0.92 MAOB (0.37) MCHR1MAOBSIGMAR1USP2POLB
SCHEMBL4394210 0.92 MCHR1 (0.34) MCHR1MAOBADRB2ADRB1ADRB3
SCHEMBL4399337 0.92 MAOB (0.41) MCHR1MAOBADRB2ADRB1ADRB3
SCHEMBL913848 0.90 KMT2A (0.38) MCHR1MAOBADRB2ADRB1ADRB3
SCHEMBL4405432 0.89 MCHR1 (0.35) MCHR1MAOBADRB2ADRB1ADRB3
SCHEMBL4401792 0.88 DRD2 (0.35) MAOBHTR1ASLC6A4TLR9TLR8
Hydrochloric Acid SCHEMBL4405309 0.88 HTR1A (0.36) MCHR1ADRB2ADRB1ADRB3HTR1A
Hydrochloric Acid SCHEMBL4405664 0.87 HTR1A (0.35) MCHR1ADRB2ADRB1ADRB3HTR1A
Hydrochloric Acid SCHEMBL4396591 0.87 HTR1A (0.34) MCHR1HTR1ASLC6A4TLR9TLR8
Hydrochloric Acid SCHEMBL4396450 0.86 SOS1 (0.36) MCHR1MAOBHTR1ASLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed