SCHEMBL4408718

SCHEMBL4408718

CC1(C)N=C(c2cnc3ccccc3c2)c2ccccc2C1(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 3/20 0.41
PDGFRA P16234 3/20 0.41
CYP2A6 P11509 1/20 0.40
BIRC5 O15392 1/20 0.39
CYP1A2 P05177 1/20 0.39
TDP2 O95551 1/20 0.39
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
NR2F2 P24468 1/20 0.38
MAP4K4 O95819 1/20 0.38
CSNK1G2 P78368 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
MAP4K5 Q9Y4K4 1/20 0.38
AKR1C3 P42330 2/20 0.37
AKR1C2 P52895 2/20 0.37
BRD4 O60885 2/20 0.37
CREBBP Q92793 2/20 0.37
NISCH Q9Y2I1 1/20 0.36
CA12 O43570 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29353363 1.00 PDGFRB (0.41) PDGFRBPDGFRACYP2A6BIRC5CYP1A2
SCHEMBL29352059 1.00 PDGFRB (0.41) PDGFRBPDGFRACYP2A6BIRC5CYP1A2
SCHEMBL4528138 0.89 NPC1 (0.40) PDGFRBPDGFRACYP2A6BIRC5CYP1A2
SCHEMBL15911291 0.89 PDGFRB (0.40) PDGFRBPDGFRAPIK3CDPIK3CAAKR1C3
SCHEMBL4523245 0.89 AKR1C3 (0.40) PDGFRBPDGFRACYP2A6BIRC5CYP1A2
SCHEMBL20521243 0.88 AKR1C3 (0.37) PDGFRBPDGFRACYP2A6BIRC5TDP2
SCHEMBL20010468 0.88 PDGFRB (0.44) PDGFRBPDGFRACYP2A6BIRC5CYP1A2
SCHEMBL4526584 0.88 CYP1A2 (0.41) PDGFRBPDGFRACYP2A6BIRC5CYP1A2
SCHEMBL4531039 0.87 BIRC5 (0.46) PDGFRBPDGFRACYP2A6BIRC5CYP1A2
SCHEMBL4524039 0.87 BIRC5 (0.46) PDGFRBPDGFRACYP2A6BIRC5CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1747 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026105160-A1 NOVEL AGROCHEMICAL COMPOSITION COMPRISING 3-SUBSTITUTED PHENYLAMIDINE COMPOUNDS AND USE THEREOF PI INDUSTRIES LTD. (IN) 2026-05-21 WO claimed
EP-4114183-B1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2026-02-25 EP claimed
US-12336537-B2 Fungicidal compositions SYNGENTA CROP PROTECTION AG (CH) 2025-06-24 US claimed
US-12310365-B2 Plant disease control composition and method for controlling plant disease by applying the same MITSUI CHEMICALS CROP & LIFE SOLUTIONS, INC. (JP) 2025-05-27 US claimed
US-20250098677-A1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2025-03-27 US claimed
US-20250040552-A1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2025-02-06 US claimed
US-20240284908-A1 Fungicidal Compositions SYNGENTA PARTICIPATIONS AG (CH) 2024-08-29 US claimed
US-11974572-B2 Fungicidal compositions SYGENTA PARTICIPATIONS AG (CH) 2024-05-07 US claimed
US-20240065267-A1 PLANT DISEASE CONTROL COMPOSITION AND METHOD FOR CONTROLLING PLANT DISEASE BY APPLYING THE SAME MITSUI CHEMICALS CROP & LIFE SOLUTIONS, INC. (JP) 2024-02-29 US claimed
US-20230413824-A1 AGROCHEMICAL COMPOSITION COMPRISING 3-SUBSTITUTED PHENYLAMIDINE COMPOUNDS AND USE THEREOF PI INDUSTRIES LTD. (IN) 2023-12-28 US claimed
WO-2014033240-A1 USE OF AN AGROCHEMICAL COMPOSITION WITH FUNGICIDAL, HERBICIDAL AND PLANT HEALTH IMPROVING ACTION IN RICE BASF SE (DE) 2014-03-06 WO claimed
EP-1736471-B1 3-(DIHYDRO(TETRAHYDRO)ISOQUINOLIN-1-YL)QUINOLINES MITSUI CHEMICALS AGRO INC (JP) 2014-01-08 EP claimed
EP-2103214-B1 USE OF QUINOLINE COMPOUNDS OR SALTS THEREOF AS ACTIVE INGREDIENTS IN SOIL- OR SEED-TREATING AGENTS AND METHOD FOR CONTROL OF PLANT DISEASE MITSUI CHEMICALS AGRO INC (JP) 2013-10-23 EP claimed
US-20120282349-A1 PLANT DISEASE CONTROL COMPOSITION AND METHOD FOR CONTROLLING PLANT DISEASE BY APPLYING THE SAME MITSUI CHEMICALS AGRO, INC. (JP) 2012-11-08 US claimed
EP-2517562-A1 PLANT DISEASE CONTROL COMPOSITION AND METHOD FOR CONTROLLING PLANT DISEASES BY APPLYING THE COMPOSITION Mitsui Chemicals Agro, Inc. (JP) 2012-10-31 EP claimed
US-20090325998-A1 SOIL TREATING AGENT OR SEED TREATING AGENT COMPRISING QUINOLINE COMPOUNDS OR SALTS THEREOF AS ACTIVE INGREDIENT,OR METHOD FOR PREVENTING PLANT DISEASES BY USING THE SAME MITSUI CHEMICALS CROP & LIFE SOLUTIONS, INC. (JP) 2009-12-31 US claimed
US-7632783-B2 fungicides, pesticides for protecting rice crop, tomatoes, cucumbers and green beans; 3-(5-fluoro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)quinoline MITSUI CHEMICALS AGRO, INC. (JP) 2009-12-15 US claimed
EP-2103214-A1 SOIL- OR SEED-TREATING AGENT COMPRISING QUINOLINE COMPOUND OR SALT THEREOF AS ACTIVE INGREDIENT, OR METHOD FOR CONTROL OF PLANT DISEASE USING THE SAME Sankyo Agro Company, Limited (JP) 2009-09-23 EP claimed
US-20080275242-A1 3-(Dihydro(Tetrahydro)Isoquinolin-1-Yl)Quinoline Compound MITSUI CHEMICALS CROP & LIFE SOLUTIONS, INC. (JP) 2008-11-06 US claimed
EP-1736471-A1 3-(DIHYDRO(TETRAHYDRO)ISOQUINOLIN-1-YL)QUINOLINES Sankyo Agro Company, Limited (JP) 2006-12-27 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250040552-A1 FUNGICIDAL COMPOSITIONS CYP51A1, CYP4X1, CYP1B1 PDGFRB 4247/4885PDGFRA 4505/4885CYP2A6 139/4885
US-20240284908-A1 Fungicidal Compositions CYP51A1, CYP4X1, CYP1B1 PDGFRB 4247/4885PDGFRA 4505/4885CYP2A6 139/4885
US-20240065267-A1 PLANT DISEASE CONTROL COMPOSITION AND METHOD FOR CONTROLLING PLANT DISEASE BY APPLYING THE SAME SNX1, HAX1, BROX PDGFRB 3596/4885PDGFRA 4203/4885CYP2A6 3516/4885
US-20230413824-A1 AGROCHEMICAL COMPOSITION COMPRISING 3-SUBSTITUTED PHENYLAMIDINE COMPOUNDS AND USE THEREOF CBR3, PFAS, PAH PDGFRB 2040/4885PDGFRA 2163/4885CYP2A6 540/4885
US-12310365-B2 Plant disease control composition and method for controlling plant disease by applying the same SNX1, HAX1, BROX PDGFRB 3596/4885PDGFRA 4203/4885CYP2A6 3516/4885
US-20080275242-A1 3-(Dihydro(Tetrahydro)Isoquinolin-1-Yl)Quinoline Compound QTRT1, RABL3, RECQL PDGFRB 4549/4885PDGFRA 4233/4885CYP2A6 995/4885
US-20120282349-A1 PLANT DISEASE CONTROL COMPOSITION AND METHOD FOR CONTROLLING PLANT DISEASE BY APPLYING THE SAME SNX1, BROX, HAX1 PDGFRB 3952/4885PDGFRA 4301/4885CYP2A6 3266/4885
US-20250098677-A1 FUNGICIDAL COMPOSITIONS CYP51A1, CYP4X1, CYP1B1 PDGFRB 4247/4885PDGFRA 4505/4885CYP2A6 139/4885
US-11974572-B2 Fungicidal compositions CYP51A1, CYP4X1, CYP1B1 PDGFRB 4247/4885PDGFRA 4505/4885CYP2A6 139/4885
US-12336537-B2 Fungicidal compositions CYP51A1, CYP4X1, CYP1B1 PDGFRB 4247/4885PDGFRA 4505/4885CYP2A6 139/4885
US-20090325998-A1 SOIL TREATING AGENT OR SEED TREATING AGENT COMPRISING QUINOLINE COMPOUNDS OR SALTS THEREOF AS ACTIVE INGREDIENT,OR METHOD FOR PREVENTING PLANT DISEASES BY USING THE SAME RABL3, H1-3, RECQL PDGFRB 2938/4885PDGFRA 2249/4885CYP2A6 829/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.