Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | HTR2A | P28223 | 9/20 | 0.40 |
| ▸ | HTR2C | P28335 | 5/20 | 0.40 |
| ▸ | HTR1A | P08908 | 4/20 | 0.40 |
| ▸ | HTR2B | P41595 | 4/20 | 0.40 |
| ▸ | SLC6A4 | P31645 | 2/20 | 0.40 |
| ▸ | HTR7 | P34969 | 2/20 | 0.40 |
| ▸ | HTR1D | P28221 | 2/20 | 0.40 |
| ▸ | HTR1B | P28222 | 2/20 | 0.40 |
| ▸ | ADRB1 | P08588 | 1/20 | 0.40 |
| ▸ | ADRA2A | P08913 | 1/20 | 0.40 |
| ▸ | SLC6A2 | P23975 | 1/20 | 0.40 |
| ▸ | HTR1E | P28566 | 1/20 | 0.40 |
| ▸ | HTR6 | P50406 | 1/20 | 0.40 |
| ▸ | SLC6A3 | Q01959 | 1/20 | 0.40 |
| ▸ | BLM | P54132 | 3/20 | 0.40 |
| ▸ | KDM4E | B2RXH2 | 2/20 | 0.40 |
| ▸ | LMNA | P02545 | 2/20 | 0.40 |
| ▸ | MAPT | P10636 | 2/20 | 0.40 |
| ▸ | TSHR | P16473 | 2/20 | 0.40 |
| ▸ | PMP22 | Q01453 | 2/20 | 0.40 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL2198661 | 0.79 | HTR2A (0.64) | HTR2AHTR2CHTR1AHTR2BSLC6A4 | |
| SCHEMBL10650990 | 0.79 | HTR2A (0.64) | HTR2AHTR2CHTR1AHTR2BSLC6A4 | |
| SCHEMBL7029247 | 0.79 | HTR2A (0.64) | HTR2AHTR2CHTR1AHTR2BSLC6A4 | |
| SCHEMBL7653075 | 0.77 | HTR2A (0.45) | HTR2AHTR2CHTR1AHTR2BSLC6A4 | |
| SCHEMBL1337678 | 0.75 | HTR1A (0.38) | HTR2AHTR2CHTR1AHTR2BSLC6A4 | |
| SCHEMBL7429865 | 0.74 | GPR84 (0.58) | HTR2AHTR2CHTR1AHTR2BSLC6A4 | |
| SCHEMBL19047013 | 0.74 | HTR2C (0.68) | HTR2AHTR2CHTR1AHTR2BSLC6A4 | |
| SCHEMBL22796513 | 0.74 | HTR2A (0.56) | HTR2AHTR2CHTR1AHTR2BSLC6A4 | |
| SCHEMBL4373291 | 0.74 | HTR2A (0.68) | HTR2AHTR2CHTR1AHTR2BSLC6A4 | |
| SCHEMBL7439210 | 0.74 | HTR2A (0.68) | HTR2AHTR2CHTR1ASLC6A4TSHR |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| WO-2011071541-A2 | CADHERIN MODULATORY AGENTS | THE SCRIPPS RESEARCH INSTITUTE (US) | 2011-06-16 | — | — | WO | claimed |
| US-9943577-B2 | Aminoacyl tRNA synthetases for modulating inflammation | ATYR PHARMA, INC. (US) | 2018-04-17 | — | — | US | disclosed |
| EP-2939689-B1 | Glutaminyl tRNA synthetases for use in the treatment of inflammatory disorders | ATYR PHARMA INC (US) | 2017-09-13 | — | — | EP | disclosed |
| US-20170202933-A1 | AMINOACYL TRNA SYNTHETASES FOR MODULATING INFLAMMATION | ATYR PHARMA, INC. | 2017-07-20 | — | — | US | disclosed |
| US-9540628-B2 | Aminoacyl tRNA synthetases for modulating inflammation | ATYR PHARMA, INC. (US) | 2017-01-10 | — | — | US | disclosed |
| US-9328340-B2 | Amino acyl tRNA synthetases for modulating inflammation | ATYR PHARMA, INC. (US) | 2016-05-03 | — | — | US | disclosed |
| EP-2939689-A1 | Glutaminyl tRNA synthetases for modulating inflammation | Atyr Pharma, Inc. (US) | 2015-11-04 | — | — | EP | disclosed |
| US-9127268-B2 | Aminoacyl tRNA synthetases for modulating inflammation | ATYR PHARMA, INC. (US) | 2015-09-08 | — | — | US | disclosed |
| US-20150140072-A1 | AMINOACYL TRNA SYNTHETASES FOR MODULATING INFLAMMATION | ATYR PHARMA, INC. | 2015-05-21 | — | — | US | disclosed |
| US-20150132277-A1 | Monomeric Forms of Human Aminoacyl-tRNA Synthetases Having Non-Canonical Biological Activities | SCRIPPS RESEARCH INST (US) | 2015-05-14 | — | — | US | disclosed |
| EP-2509625-B1 | HISTIDYL TRNA SYNTHETASES FOR REDUCING INFLAMMATION | ATYR PHARMA INC (US) | 2015-01-28 | — | — | EP | disclosed |
| US-8828395-B2 | Antibodies that bind tyrosyl-tRNA synthetases | ATYR PHARMA, INC. (US) | 2014-09-09 | — | — | US | disclosed |
| US-8828685-B2 | Monomeric forms of human aminoacyl-t-RNA synthetases having non-canonical biological activities | THE SCRIPPS RESEARCH INSTITUTE (US) | 2014-09-09 | — | — | US | disclosed |
| US-20130273045-A1 | AMINO ACYL TRNA SYNTHETASES FOR MODULATING INFLAMMATION | ATYR PHARMA, INC. | 2013-10-17 | — | — | US | disclosed |
| US-20130108630-A1 | AMINO ACYL TRNA SYNTHETASES FOR MODULATING INFLAMMATION | ATYR PHARMA, INC. | 2013-05-02 | — | — | US | disclosed |
| US-20130052177-A1 | MONOMERIC FORMS OF HUMAN AMINOACYL-t-RNA SYNTHETASES HAVING NON-CANONICAL BIOLOGICAL ACTIVITIES | THE SCRIPPS RESEARCH INSTITUTE (US) | 2013-02-28 | — | — | US | disclosed |
| US-20120064082-A1 | AMINOACYL TRNA SYNTHETASES FOR MODULATING HEMATOPOIESIS | ATYR PHARMA, INC. (US) | 2012-03-15 | — | — | US | disclosed |
| WO-2011097031-A2 | MONOMERIC FORMS OF HUMAN AMINOACYL-TRNA SYNTHETASES HAVING NON-CANONICAL BIOLOGICAL ACTIVITIES | THE SCRIPPS RESEARCH INSTITUTE (US) | 2011-08-11 | — | — | WO | disclosed |
| US-20110150885-A1 | AMINOACYL TRNA SYNTHETASES FOR MODULATING HEMATOPOIESIS | ATYR PHARMA, INC. (US) | 2011-06-23 | — | — | US | disclosed |
| WO-2011071541-A2 | CADHERIN MODULATORY AGENTS | THE SCRIPPS RESEARCH INSTITUTE (US) | 2011-06-16 | — | — | WO | disclosed |