SCHEMBL440988

SCHEMBL440988

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nearest known ligand 0.00

Known targets — ChEMBL curated mechanism

GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHMGCRMMP1MMP13MMP7MMP8PTGS1PTGS2ileSpolrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL438215 0.91
SCHEMBL437398 0.91
SCHEMBL437397 0.91
Zinc Ion SCHEMBL439179 0.91
SCHEMBL441708 0.91
SCHEMBL10613758 0.78
SCHEMBL1656667 0.78 CES2 (0.30)
SCHEMBL3658234 0.73 CES2 (0.39)
SCHEMBL1659521 0.70 CES2 (0.30)
SCHEMBL20985817 0.70 CES2 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230173731-A1 FLAME-RETARDANT BIAXIALLY-ORIENTED POLYESTER FILM TOYOBO CO., LTD. (JP) 2023-06-08 US disclosed
US-10208175-B2 Flame-retardant biaxially oriented polyester film, and flame-retardant polyester film laminate comprising the same and flexible circuit board TEIJIN DUPONT FILMS JAPAN LIMITED (JP) 2019-02-19 US disclosed
EP-3064549-B1 FLAME-RETARDANT BIAXIALLY-ORIENTED POLYESTER FILM, AND FLAME-RETARDANT POLYESTER FILM LAYERED BODY AND FLEXIBLE CIRCUIT BOARD COMPRISING SAME TEIJIN DUPONT FILMS JAPAN LTD (JP) 2017-11-22 EP disclosed
EP-3064549-A1 FLAME-RETARDANT BIAXIALLY-ORIENTED POLYESTER FILM, AND FLAME-RETARDANT POLYESTER FILM LAYERED BODY AND FLEXIBLE CIRCUIT BOARD COMPRISING SAME Teijin Dupont Films Japan Limited (JP) 2016-09-07 EP disclosed
US-20160194466-A1 FLAME-RETARDANT BIAXIALLY ORIENTED POLYESTER FILM, AND FLAME-RETARDANT POLYESTER FILM LAMINATE COMPRISING THE SAME AND FLEXIBLE CIRCUIT BOARD TEIJIN DUPONT FILMS JAPAN LIMITED (JP) 2016-07-07 US disclosed
US-20120064790-A1 Ethylene Diphosphinic Acids CLARIANT FINANCE (BVI) LIMITED (VG) 2012-03-15 US disclosed
EP-1967549-B1 USE OF A FLAME-RETARDANT RESIN COMPOSITION FOR TRANSMISSION SIDE MEMBER IN LASER WELDING WINTECH POLYMER LTD (JP) 2012-02-29 EP disclosed
US-8084518-B2 Ethylenebis(hydroxyalkylphosphinic acid) and salts thereof CLARIANT FINANCE (BVI) LIMITED (VG) 2011-12-27 US disclosed
EP-2081942-B1 ETHYLENE DIPHOSPHINIC ACIDS CLARIANT FINANCE BVI LTD (VG) 2011-12-14 EP disclosed
US-20100233474-A1 FLAME-RETARDANT RESIN COMPOSITION FORMING LASER-TRANSMITTABLE MEMBER WINTECH POLYMER LTD. (JP) 2010-09-16 US disclosed
US-20100093239-A1 Ethylene Diphosphinic Acids CLARIANT INTERNATIONAL LTD. (CH) 2010-04-15 US disclosed
US-7612131-B2 Flame-retardant resin composition WINTECH POLYMER LTD. (JP) 2009-11-03 US disclosed
EP-2081942-A1 ETHYLENE DIPHOSPHINIC ACIDS Clariant Finance (BVI) Limited (VG) 2009-07-29 EP disclosed
EP-1967549-A1 FLAME-RETARDANT RESIN COMPOSITION FOR TRANSMISSION SIDE MEMBER IN LASER WELDING Wintech Polymer Ltd. (JP) 2008-09-10 EP disclosed
US-20080167406-A1 FLAME-RETARDANT RESIN COMPOSITION WINTECH POLYMER, LTD. (JP) 2008-07-10 US disclosed
EP-1935944-A2 Flame-retardant resin composition Wintech Polymer Ltd. (JP) 2008-06-25 EP disclosed
WO-2008043499-A1 ETHYLENE DIPHOSPHINIC ACIDS CLARIANT FINANCE (BVI) LIMITED (VG) 2008-04-17 WO disclosed