SCHEMBL4410091

SCHEMBL4410091

COc1cc(C(C)=O)cc2[nH]ncc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.50
METAP2 P50579 4/20 0.45
CYP1A2 P05177 2/20 0.45
ACACB O00763 1/20 0.42
ACACA Q13085 1/20 0.42
MAOB P27338 3/20 0.40
BRD4 O60885 1/20 0.40
AXL P30530 1/20 0.40
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
TDO2 P48775 1/20 0.38
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
TYK2 P29597 1/20 0.38
JAK3 P52333 1/20 0.38
MAOA P21397 1/20 0.38
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2671673 0.88 CA12 (0.50) METAP2CYP1A2ACACBACACAMAOB
SCHEMBL1722163 0.86 TDO2 (0.50) METAP2CYP1A2ACACBACACAMAOB
SCHEMBL4137015 0.84 METAP2 (0.45) METAP2CYP1A2ACACBACACAMAOB
SCHEMBL4407859 0.84 METAP2 (0.42) METAP2CYP1A2ACACBACACAMAOB
SCHEMBL1723345 0.81 HSD17B2 (0.49) LMNAMETAP2CYP1A2SMN1; SMN2TDO2
SCHEMBL17277752 0.78 NOS1 (0.43) METAP2MAOBROCK2ROCK1JAK2
SCHEMBL24656061 0.73 AXL (0.44) METAP2CYP1A2BRD4AXLROCK2
SCHEMBL2008097 0.73 IDO1 (0.56) METAP2CYP1A2BRD4AXLTDO2
SCHEMBL29990549 0.73 IDO1 (0.56) METAP2CYP1A2BRD4AXLTDO2
SCHEMBL31411282 0.73 METAP2 (0.49) METAP2CYP1A2BRD4AXLTDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012056372-A1 N1/N2-LACTAM ACETYL-CoA CARBOXYLASE INHIBITORS PFIZER INC. (US) 2012-05-03 WO disclosed